Abstract
2-Phenyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimtdine-5,7-dione reacts with several nucleophilc reagents via a scheme involving nucleophilic addition with opening of the dioxopyrimidine ring at the C-N bond in the 7–8 positions. The reaction may serve as a method for the synthesis of some asymmetrical pyrazolyl derivatives of malonic acid.
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See [1] for communication I.
Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 8, pp. 1145–1147, August, 1971.
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Dashkevich, L.B., Samoletov, M.M. & Tkachenko, M.L. Investigation of condensed heterocyclic pyrimido systems. Chem Heterocycl Compd 7, 1077–1079 (1971). https://doi.org/10.1007/BF00477402
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DOI: https://doi.org/10.1007/BF00477402