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Efficient Synthesis of Highly Functionalized Thiazolidine-4-ones Under Solvent-Free Conditions

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Summary.

4-Phenylthiosemicarbazide reacts smoothly with dimethyl acetylenedicarboxylate in the presence of aldehydes or ketones under solvent free conditions to produce highly functionalized thiazolidine-4-ones.

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Authors and Affiliations

  1. Chemistry Department, Tarbiat Modares University, Tehran, Iran

    Issa Yavari, Nargess Hosseini & Loghman Moradi

Authors
  1. Issa Yavari
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  2. Nargess Hosseini
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  3. Loghman Moradi
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Correspondence to Issa Yavari.

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Yavari, I., Hosseini, N. & Moradi, L. Efficient Synthesis of Highly Functionalized Thiazolidine-4-ones Under Solvent-Free Conditions. Monatsh Chem 139, 133–136 (2008). https://doi.org/10.1007/s00706-007-0751-x

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  • DOI: https://doi.org/10.1007/s00706-007-0751-x

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