1. Synthetic coumarin derivatives with anticoagulation and antiplatelet aggregation inhibitory effects

   • Triveena M. Ramsis
   • Maha A. Ebrahim
   • Eman A. Fayed

   Review Article Open access 16 September 2023 Pages: 2269 - 2278

   

2. Advances in research of ursolic acid and its derivatives as potential drug candidates against various types of lung cancers

   • Li Song
   • Ling Dai
   • Xing Zheng

   Review Article 25 September 2023 Pages: 2279 - 2298

   

3. Structural and stereochemical determinants for hGAT3 inhibition: development of novel conformationally constrained and substituted analogs of (S)-isoserine

   • F. Bavo
   • S. Kickinger
   • B. Frølund

   Original Research Article Open access 16 August 2023 Pages: 2299 - 2324

   

4. Synthesis of berberine derivatives and their antiviral activity toward respiratory syncytial virus

   • Anna A. Shtro
   • Elizaveta D. Gladkova
   • Nariman F. Salakhutdinov

   Original Research Article 18 August 2023 Pages: 2325 - 2333

   

5. New tolfenamic acid derivatives with hydrazine-1-carbothioamide and 1,3,4-oxadiazole moieties targeting VEGFR: synthesis, in silico studies, and in vitro anticancer assessment

   • Abbas A. Ridha Mehihi
   • Ammar A. Razzak Kubba
   • Lubna H. Tahtamouni

   Original Research Article 18 August 2023 Pages: 2334 - 2348

   

6. Bioactivity-guided isolation of anti-acetylcholinesterase compounds from Odontites vulgaris Moench

   • Liang Liu
   • Xuejian Chang
   • Xianwen Zhang

   Original Research Article 19 August 2023 Pages: 2349 - 2355

   

7. Molecular modeling of the phosphoglycerate kinase and fructose-bisphosphate aldolase proteins from Candida glabrata and Candida albicans

   • Nancy A. Vázquez-López
   • Rodrigo Aguayo-Ortiz
   • Mayra Cuéllar-Cruz

   Original Research Article 19 August 2023 Pages: 2356 - 2369

   

8. Influence of alkyl linkers on the anti-breast cancer activity of dihydroartemisinin-isatin hybrids

   • Yang Xie
   • Kai Zhang
   • Xiangyang Sun

   Original Research 21 August 2023 Pages: 2370 - 2375

   

9. Ester tethered artemisinin-isatin hybrids: design, synthesis and anti-leukemic activity evaluation

   • Peng Wang
   • Dai Yuan
   • Li Kong

   Original Research 21 August 2023 Pages: 2376 - 2379

   

10. Bio-evaluation of the 2-nitrochalcones as potential anti-lung cancer agents, inducers of apoptosis and inhibitors of protein kinase (VEGFR-2)

    • Malose J. Mphahlele
    • Garland K. More
    • Yee Siew Choong

    Original Research Article Open access 29 August 2023 Pages: 2380 - 2393

    

11. Synthesis, anticancer evaluation and docking studies of novel adamantanyl-1,3,4-oxadiazol hybrid compounds as Aurora-A kinase inhibitors

    • Areej M. Jaber
    • Mohammed M. Al-Mahadeen
    • Mutasem O. Taha

    Original Research Article 06 September 2023 Pages: 2394 - 2404

    

12. Synthesis, in silico, and evaluation of AChE inhibitory activity of N-phthaloylphenylglycine derivatives as potential anti-Alzheimer’s agents

    • Erik Andrade-Jorge
    • Natalia Reyes-Vallejo
    • Adelfo Reyes-Ramírez

    Original Research Article Open access 09 September 2023 Pages: 2405 - 2418

    

13. Synthesis, in-silico based virtual screening,anti-cancer potential of novel1,2,3-triazole-thiadiazole hybrid derivatives as Aurora kinase A (ARK-A) and Extracellular regulated kinase 2 (ERK2) dual inhibitors

    • Lingaiah Bontha
    • Praveen Kumar Edigi
    • Satyanarayana Sirasani

    Original Research Article 12 September 2023 Pages: 2419 - 2431

    

14. Design, synthesis and antiproliferative activity of ACY-1215 analogs as potent selective histone deacetylases 6 inhibitors

    • Hongfei Duan
    • Jiayun Wang
    • Xinyang Chen

    Original Research Article 20 September 2023 Pages: 2432 - 2441