Alkaloids derived from the genus Daphniphyllum Xu LiangXin-Zhou YangJing-Quan Yuan Review Article 13 October 2020 Pages: 1 - 14
The novel scaffold 1,2,4-benzothiadiazine-1,1-dioxide: a review Sumit ChhabraKamal Shah Review Article 14 October 2020 Pages: 15 - 30
Pyrimidine and fused pyrimidine derivatives as promising protein kinase inhibitors for cancer treatment Khaled R. A. AbdellatifRania B. Bakr Review Article 29 October 2020 Pages: 31 - 49
Tankyrase inhibitors: emerging and promising therapeutics for cancer treatment Anu VermaAshwani KumarParvin Kumar Review Article 17 November 2020 Pages: 50 - 73
Synthesis and anticancer evaluation of amide derivatives of imidazo-pyridines Chekuri Sharmila RaniAlugubelli Gopi ReddyMandava Venkata Basaveswara Rao Original Research 01 October 2020 Pages: 74 - 83
Synthesis of novel selenotetrazole purine derivatives and their potential chemotherapeutic activities Gulay DilekIshak Ozel TekinZuhal Gercek Original Research 02 October 2020 Pages: 84 - 97
First in class (S,E)-11-[2-(arylmethylene)hydrazono]-PBD analogs as selective CB2 modulators targeting neurodegenerative disorders David MingleMeirambek OspanovMohamed A. Ibrahim Original Research 04 October 2020 Pages: 98 - 108
Synthesis, characterization and antimalarial activity of isoquinoline derivatives Sewan TheeramunkongArtitiya ThiengsusukPhunuch Muhamad Original Research 06 October 2020 Pages: 109 - 119
Dihydropyrimidones: A ligands urease recognition study and mechanistic insight through in vitro and in silico approach Farman Ali KhanShahbaz ShamimAjmal Khan Original Research 06 October 2020 Pages: 120 - 132
Structure-based design, synthesis, biological evaluation, and molecular docking of novel 10-methoxy dibenzo[b,h][1,6]naphthyridinecarboxamides K. N. VennilaB. SelvakumarK. P. Elango Original Research 11 October 2020 Pages: 133 - 141
Synthesis and antitumor effects of a new class of 1,2,4-triazole derivatives Zheng WuXin LiBao-Quan Chen Original Research 19 October 2020 Pages: 142 - 151
Antimicrobial and antileishmanial activities of extracts and some constituents from the leaves of Solanum chrysotrichum Schldl Guillermo Núñez-MojicaVerónica M. Rivas-GalindoMaría del Rayo Camacho-Corona Original Research 21 October 2020 Pages: 152 - 162
A facile synthesis of some new pyrimidine-2,4,6-triones analogs and their O-β-D-glucosides P-glycoprotein and antioxidant, antimicrobial study, blood–brain barrier, cytochrome p450 enzyme activity prediction Kishor M. HatzadeAjay M. GhatoleGunwant P. Gadekar Original Research 22 October 2020 Pages: 163 - 181
Design, synthesis and effect of triazole derivatives against some toxic activities of Bothrops jararaca venom Aldo R. da SilvaAna Cláudia R. da SilvaAndré L. Fuly Original Research 22 October 2020 Pages: 182 - 195
First-time comparative investigation on Araucaria columnaris (G. Forst.) Hook. leaves: extraction techniques, phytochemicals, medicinal activities, and DFT study Poonam K. PatialDamanjit S. Cannoo Original Research 27 October 2020 Pages: 196 - 214
A simple model for the assessment of the agonistic activity of dibenzazepine derivatives by molecular moieties Mohammad Hossein KeshavarzHossein FakhraianNorollah Saedi Original Research 30 October 2020 Pages: 215 - 225
Synthesis, urease inhibition screening and molecular docking studies of piperonal based imine derivatives Obaid-ur-Rahman AbidSaima DaudMuhammad Yasir Original Research 31 October 2020 Pages: 226 - 235
Novel approach of multi-targeted thiazoles and thiazolidenes toward anti-inflammatory and anticancer therapy—dual inhibition of COX-2 and 5-LOX enzymes Jaismy Jacob PManju S L Original Research 01 November 2020 Pages: 236 - 257
Potent antiproliferative active agents: novel bis Schiff bases and bis spiro β-lactams bearing isatin tethered with butylene and phenylene as spacer and DNA/BSA binding behavior as well as studying molecular docking Mohammad BashiriAliasghar JarrahpourEdward Turos Original Research 11 November 2020 Pages: 258 - 284
Design, synthesis, and evaluation of different scaffold derivatives against NS2B-NS3 protease of dengue virus Lata R. GanjiLekha GandhiMeena A. Kanyalkar Original Research 17 November 2020 Pages: 285 - 301