1. New Delhi metallo-β-lactamase-1 inhibitors for combating antibiotic drug resistance: recent developments

   • Ajmer Singh Grewal
   • Komal Thapa
   • Sukhbir Singh

   Review Article 10 June 2020 Pages: 1301 - 1320

   

2. Synthesis and biological evaluation of α- and β-hydroxy substituted amino acid derivatives as potential mGAT1–4 inhibitors

   • Janina C. Andreß
   • Michael C. Böck
   • Klaus T. Wanner

   Original Research Open access 08 May 2020 Pages: 1321 - 1340

3. Synthesis and antitumor activity of novel gibberellin derivatives with tetracyclic diterpenoid skeletons

   • Shi-ying Zhu
   • Fa-zeng Luo
   • Ping-Hua Sun

   Original Research 09 May 2020 Pages: 1341 - 1354

   

4. Cytotoxicity, anticancer, and antioxidant properties of mono and bis-naphthalimido β-lactam conjugates

   • Nassim Borazjani
   • Maryam Behzadi
   • Edward Turos

   Original Research 10 May 2020 Pages: 1355 - 1375

   

5. Synthesis and biological evaluation of novel N-2,4-dimethoxyphenyl dithiolopyrrolone derivatives as bacterial RNA polymerase inhibitors

   • Jieyun Meng
   • Bo Kong
   • Xiangduan Tan

   Original Research 12 May 2020 Pages: 1376 - 1386

   

6. Synthesis and in vitro antimycobacterial and antileishmanial activities of hydroquinone-triazole hybrids

   • Chris-Marie Horn
   • Janine Aucamp
   • David D. N’Da

   Original Research 12 May 2020 Pages: 1387 - 1399

   

7. Synthesis of 1-(4-hydroxy-3-methoxyphenyl)-2,3,4,9-tetrahydro-1H-β-carboline-3-carboxylic acid derivatives as mast cell stabilizers

   • Karan Saini
   • Jatinder Singh
   • Ram Sarup Singh

   Original Research 12 May 2020 Pages: 1400 - 1412

   

8. Synthesis and biological evaluation of a new series of 1-aryl-3-[4-(pyridin-2-ylmethoxy)phenyl]urea derivatives as new anticancer agents

   • Jian Feng
   • Tai Li
   • Chun Hu

   Original Research 18 May 2020 Pages: 1413 - 1423

   

9. Synthesis and evaluation of substituted phenyl cycloalkylureas and bioisosteres as IL-6 expression inhibitors

   • Sébastien Tremblay
   • Joël Boutin
   • René C.-Gaudreault

   Original Research 19 May 2020 Pages: 1424 - 1437

   

10. Design, synthesis, and biological evaluation of novel benzo[b]thiophene-diaryl urea derivatives as potential anticancer agents

    • Omid Zarei
    • Fereshteh Azimian
    • Siavoush Dastmalchi

    Original Research 19 May 2020 Pages: 1438 - 1448

    

11. Synthesis and biological evaluation of selected 7-azaindole derivatives as CDK9/Cyclin T and Haspin inhibitors

    • Lianie Pieterse
    • Lesetja J. Legoabe
    • Sandrine Ruchaud

    Original Research 22 May 2020 Pages: 1449 - 1462

    

12. Discovery of anti-influenza nucleoside triphosphates targeting the catalytic site of A/PR/8/34/H1N1 polymerase

    • Nataraj Sekhar Pagadala
    • Rakesh Bhat
    • Abdolamir Landi

    Original Research 24 May 2020 Pages: 1463 - 1477

    

13. Evaluation of cholinesterase inhibitory activity and cytotoxicity of synthetic derivatives of di- and triterpene metabolites from Pinus silvestris and Dipterocarpus alatus resins

    • Irina E. Smirnova
    • Oxana B. Kazakova
    • Rene Csuk

    Original Research 31 May 2020 Pages: 1478 - 1485

    

14. Efficient synthesis of 2,3-diarylbenzo[b]thiophene molecules through palladium (0) Suzuki–Miyaura cross-coupling reaction and their antithrombolyitc, biofilm inhibition, hemolytic potential and molecular docking studies

    • Nosheen Sial
    • Nasir Rasool
    • Syed Adnan Ali Shah

    Original Research 02 June 2020 Pages: 1486 - 1496

    

15. Cytotoxic, anti-inflammatory, and α-glucosidase inhibitory effects of flavonoids from Lippia graveolens (Mexican oregano)

    • Sonia Amador
    • Antonio Nieto-Camacho
    • Emma Maldonado

    Original Research 02 June 2020 Pages: 1497 - 1506

    

16. Synthesis, evaluation of cytotoxicity, and antimicrobial activity of A-azepano- and A-seco-3-amino-C28-aminolupanes

    • Oxana B. Kazakova
    • Tatyana V. Lopatina
    • Kyrill Yu. Suponitsky

    Original Research 07 June 2020 Pages: 1507 - 1519

    

17. Synthesis and antiseizure activity of (E)-1,2-diarylethylidenehydrazine carboximidamides against tonic-clonic seizures: an intracerebroventricular and electrophysiological study

    • Fariba Abedi Firouzjaei
    • Elmira Heidarli
    • Hamid Irannejad

    Original Research 09 June 2020 Pages: 1520 - 1535

    

18. Uses of dimedone to synthesis pyrazole, isoxazole and thiophene derivatives with antiproliferative, tyrosine kinase and Pim-1 kinase inhibitions

    • Rafat Milad Mohareb
    • Fatma Mohamed Manhi
    • Amal Abdelwahab

    Original Research 12 June 2020 Pages: 1536 - 1551