Natural thiopeptides as a privileged scaffold for drug discovery and therapeutic development Xiaoqi ShenMuhammad MustafaJiangtao Gao Review Article 29 May 2019 Pages: 1063 - 1098
Sulfa drug analogs: new classes of N-sulfonyl aminated azines and their biological and preclinical importance in medicinal chemistry (2000–2018) Galal H. ElgemeieRasha A. AzzamRasha E. Elsayed Review Article 12 June 2019 Pages: 1099 - 1131
Synthesis, molecular docking, and apoptogenic efficacy of novel N-heterocycle analogs to target B-cell lymphoma 2/X-linked inhibitors of apoptosis proteins to regress melanoma Zabiulla ZabiullaVikas H. MalojiraoShaukath Ara Khanum Original Research 04 June 2019 Pages: 1132 - 1160
Umbelliferone isolated from Zosima absinthifolia roots partially restored erectile dysfunction in streptozotocin-induced diabetic rats Songul KarakayaDidem Yilmaz-OralSerap Gur Original Research 31 May 2019 Pages: 1161 - 1167
Quinoline analogs of 2-aminoindane as potential central dopaminergic agents Jorge E. AngelRicardo D. EnrizSebastian A. Andujar Original Research 30 May 2019 Pages: 1168 - 1181
Synthesis and in vitro evaluation of substituted tetrahydroquinoline-isoxazole hybrids as anticancer agents Fausto M. GüizaYenny Bueno DuarteArnold R. Romero Bohórquez Original Research 01 June 2019 Pages: 1182 - 1196
Functional relaxant effect of 6,7-dipropoxy-2H-chromen-2-one is mainly by calcium channel blockade in ex vivo assay of tracheal rings Amanda Sánchez-RecillasSamuel Estrada-SotoItzell A. Gallardo-Ortiz Original Research 31 May 2019 Pages: 1197 - 1204
In vitro activity of novel derivatives of 1,3-oxazole-4-carboxylate and 1,3-oxazole-4-carbonitrile against human cytomegalovirus Maryna V. KachaevaStepan G. PilyoVolodymyr S. Brovarets Original Research 31 May 2019 Pages: 1205 - 1211
Synthesis of oleanolic acid/ursolic acid/glycyrrhetinic acid-hydrogen sulfide donor hybrids and their antitumor activity Li-xin ShengJia-yan HuangKe-guang Cheng Original Research 04 June 2019 Pages: 1212 - 1222
Green synthesis and 3D pharmacophore study of pyrimidine and glucoside derivatives with in vitro potential anticancer and antioxidant activities Mounir A. SalemMohamed S. BehaloEman Elrazaz Original Research 31 May 2019 Pages: 1223 - 1234
Pyrazole–chalcone derivatives as selective COX-2 inhibitors: design, virtual screening, and in vitro analysis Anelise F. MacariniThales U. C. SobrinhoRogério Corrêa Original Research 30 May 2019 Pages: 1235 - 1245
3D-QSAR, molecular docking, and new compound design of pyrimidine derivatives as Src small molecule inhibitors Jun-wei WangYa-ting DengZhi-hua Lin Original Research 05 June 2019 Pages: 1246 - 1263
Antiplatelet activity and TNF-α release inhibition of phthalimide derivatives useful to treat sickle cell anemia Rafael C. ChelucciIsabela J. de OliveiraManChin Chung Original Research 31 May 2019 Pages: 1264 - 1271
New fluoroquinolones/nitric oxide donor hybrids: design, synthesis and antitubercular activity Hossameldin A. AzizGamal A. I. MoustafaGamal El-Din A. Abuo-Rahma Original Research 06 June 2019 Pages: 1272 - 1283
Design, synthesis, biological evaluation and molecular modeling of new coumarin derivatives as potent anticancer agents Eman A. FayedRehab SabourAhmed B. M. Mehany Original Research 01 June 2019 Pages: 1284 - 1297
Preparation and biological evaluation of quinoline amines as anticancer agents and its molecular docking Kailasam N. VennilaKolandhaivel PrabhaKuppannagounder P. Elango Original Research 01 June 2019 Pages: 1298 - 1307
A structure–activity relationship study of phenyl sesquiterpenoids on efflux inhibition against Staphylococcus aureus Zhong-Lin SunTao LiuQing Mu Original Research 06 June 2019 Pages: 1308 - 1318
Fluorophenols bearing nitrogenated heterocycle moieties, a class of novel Keap1-Nrf2 protein-protein interaction inhibitors: synthesis, antioxidant stress screening and molecular docking Xiu E FengDe Peng KongQing Shan Li Original Research 06 June 2019 Pages: 1319 - 1337