Quinazolines as inhibitors of chromatin-associated proteins in histones Frida S. Herrera-VázquezFrancisco Hernández-LuisJosé L. Medina Franco Review Article 04 February 2019 Pages: 395 - 416
Developmental perspectives of the drugs targeting enzyme-instigated inflammation: a mini review Parteek PrasherHarish MudilaBeena Khati Review Article 02 March 2019 Pages: 417 - 449
Effect of chiral polyhydrochromenes on cannabinoid system Nikolai S. Li-ZhulanovIrina V. Il’inaNariman F. Salakhutdinov Original Research 01 February 2019 Pages: 450 - 464
Design, synthesis and anticancer activities of halogenated Phenstatin analogs as microtubule destabilizing agent Shengquan HuWuji SunHong Yan Original Research 04 February 2019 Pages: 465 - 472
Total synthesis of the linear and angular 3-methylated regioisomers of the marine natural product Kealiiquinone and biological evaluation of related Leucetta sp. alkaloids on human breast cancer César R. Solorio-AlvaradoVelayudham RamadossAngel J. Alonso-Castro Original Research 08 February 2019 Pages: 473 - 484
New indole and indazole derivatives as potential antimycobacterial agents Violina T. AngelovaTania PenchevaVioleta Valcheva Original Research 08 February 2019 Pages: 485 - 497
4D-QSAR studies of CB2 cannabinoid receptor inverse agonists: a comparison to 3D-QSAR Houpan ZhangQiaoli LvGuogang Tu Original Research 11 February 2019 Pages: 498 - 504
LC-MS-based metabolomic profiling of Lepidium coronopus water extract, anti-inflammatory and analgesic activities, and chemosystematic significance Ahmed ElkhateebMona El-ShabrawySameh R. Hussein Original Research 14 February 2019 Pages: 505 - 514
Chemical composition, antioxidant, anti-lipooxygenase, antimicrobial, anti-parasite and cytotoxic activities of Polyalthia longifolia seed oil O. AtolaniE. T. ArehG. A. Olatunji Original Research 22 February 2019 Pages: 515 - 527
Nano Sb2O3 catalyzed green synthesis, cytotoxic activity, and molecular docking study of novel α-aminophosphonates Sreelakshmi PoolaMaheshwara Reddy NadiveedhiSuresh Reddy Cirandur Original Research 23 February 2019 Pages: 528 - 544
Design, synthesis, cytotoxicity, and molecular modeling study of 2,4,6-trisubstituted pyrimidines with anthranilate ester moiety Kirill P. CheremnykhVictor A. SavelyevElvira E. Shults Original Research 23 February 2019 Pages: 545 - 558
Design, synthesis and molecular docking studies of quinazolin-4-ones linked to 1,2,3-triazol hybrids as Mycobacterium tuberculosis H37Rv inhibitors besides antimicrobial activity Narendra Kumar MaddaliI. V. Kasi Viswanath*Vanajakshi Gudla Original Research 04 March 2019 Pages: 559 - 570
Synthesis and in vitro biological evaluation of 1,3-bis-(1,2,3-triazol-1-yl)-propan-2-ol derivatives as antifungal compounds fluconazole analogues Armando Zambrano-HuertaDamián David Cifuentes-CastañedaErick Cuevas-Yañez Original Research 09 March 2019 Pages: 571 - 579
Synthesis and anticancer activity evaluation of novel oxacalix[2]arene[2]pyrimidine derivatives Tonghui HuangXin WuXiaoxing Yin Original Research 11 March 2019 Pages: 580 - 590
Xenicanes attenuate pro-inflammatory 5-lipoxygenase: Prospective natural anti-inflammatory leads from intertidal brown seaweed Padina tetrastromatica Tima AntonyKajal Chakraborty Original Research 11 March 2019 Pages: 591 - 607
Furanchalcone–biphenyl hybrids: synthesis, in silico studies, antitrypanosomal and cytotoxic activities Elisa GarcíaRodrigo OchoaWilson Cardona-G Original research 11 March 2019 Pages: 608 - 622