Inhibitor discovery from pomegranate rind for targeting human salivary α-amylase Jiachen SunShengjie DongWenyuan Gao Original Research 17 April 2018 Pages: 1559 - 1577
Methotrexate-conjugated to polymer quantum dot for cytotoxicity effect improved against MCF-7 and Hela cells Mohammad RafieniaVahid NasirianAsad Vaisi-Raygani Original Research 28 March 2018 Pages: 1578 - 1588
Spectroscopic investigation on the interaction characteristics and inhibitory activities between baicalin and acetylcholinesterase Mingyan SunMing SuHanwen Sun Original Research 20 April 2018 Pages: 1589 - 1598
Synthesis, evaluation, and molecular properties prediction of substituted cinnamoylpiperazine derivatives as potential antinociceptive and anticonvulsive agents Gummalla PrasanthiKvsrg PrasadKoganti Bharathi Original Research 07 April 2018 Pages: 1599 - 1608
Synthesis of asiatic acid derivatives and their cytotoxic activity Loc Tran VanQuynh Nhu Vo ThiSung Tran Van Original Research 06 April 2018 Pages: 1609 - 1623
Synthesis, antimicrobial activity, and molecular docking study of fluorine-substituted indole-based imidazolines Humberto L. Mendoza-FigueroaMaria Trinidad Serrano-AlvaMartha S. Morales-Ríos Original Research 06 April 2018 Pages: 1624 - 1633
Dual targeting agents for Aβ plaque/P-glycoprotein and Aβ plaque/nicotinic acetylcholine α4β2* receptors—potential approaches to facilitate Aβ plaque removal in Alzheimer’s disease brain Gurleen K. SamraKenneth DangJogeshwar Mukherjee Original Research 07 April 2018 Pages: 1634 - 1646
Synthesis, X-ray crystallographic study, pharmacology and docking of hydrazinyl thiazolyl coumarins as dengue virus NS2B/NS3 serine protease inhibitors Samina Khan YusufzaiHasnah OsmanIbrahim Abdul Razak Original Research 20 April 2018 Pages: 1647 - 1665
Selective and novel cyclin-dependent kinases 4 inhibitor: synthesis and biological evaluation Qingxiang GuoYongtao LiYan Fan Original Research 20 April 2018 Pages: 1666 - 1678
Oxygenated heterocyclic metabolites with dual cyclooxygenase-2 and 5-lipoxygenase inhibitory potentials from Rhizophora annamalayana Kajal ChakrabortyVamshi Krishna Raola Original Research 04 May 2018 Pages: 1679 - 1689
Synthesis of new C-dimethylated chalcones as potent antitubercular agents Rambabu AnandamSurender Singh JadavHari Babu Bollikolla Original Research 04 May 2018 Pages: 1690 - 1704
Structural characterization, biochemical, inhibition and computational studies of Entamoeba histolytica phosphoglycerate mutase: finding hits for a new antiamoebic drug Artemisa Luévano-De la CruzElkin Eduardo Sanabria-ChanagaAlfredo Téllez-Valencia Original Research 07 May 2018 Pages: 1705 - 1716
Synthesis and evaluation of coumarin/piperazine hybrids as acetylcholinesterase inhibitors Juan ZhangCheng-Shi Jiang Original Research 04 May 2018 Pages: 1717 - 1727
New camphor hybrids: lipophilic enhancement improves antimicrobial efficacy against drug-resistant pathogenic microbes and intestinal worms Ramalingam PeramanAmit K. TiwariRaghuveer V. Pemmidi Original Research 12 May 2018 Pages: 1728 - 1739
Correction to: Cytotoxic and anti-inflammatory compounds from Red Sea grass Thalassodendron ciliatum Reda F. AbdelhameedAmany K. IbrahimSafwat A. Ahmed Publisher Correction 09 May 2018 Pages: 1740 - 1740