Synthesis of tetrahydropyrazolo-quinazoline and tetrahydropyrazolo-pyrimidocarbazole derivatives as potential anti-prostate cancer agents and Pim-1 kinase inhibitors Rafat M. MoharebNermeen S. AbbasAbeer A. Mohamed Original Research 04 March 2017 Pages: 1073 - 1088
Synthesis, characterization and antimicrobial studies on 3-((4-(4-nitrophenyl)-6-aryl-1,6-dihydropyrimidin-2-yl)thio)propanenitriles and their derivatives N. C. DesaiDarshan PandyaDarshita Vaja Original Research 04 March 2017 Pages: 1089 - 1097
Novel substituted 3-phenyl 1-(4-(5-bromopyridin-3-yl)-6-phenylpyrimidin-2-yl)-thiourea compounds as key small organic molecules for the potential treatment of type II diabetes mellitus: in vitro studies against yeast α-glucosidase Tanzeel Ur RehmanIslam Ullah KhanSadaf Riaz Original Research 06 March 2017 Pages: 1098 - 1106
Synthesis and antimicrobial activity of newly synthesized 4-substituted-pyrazolo[3,4-d]pyrimidine derivatives Ahmed M. El-SayedSamy M. IbrahimMansour E. Abo-Kul Original Research 06 March 2017 Pages: 1107 - 1116
Iridoid and phenylpropanoid glycosides from the roots of Lantana montevidensis Nesma M. MohamedMakboul A. MakboulSamir A. Ross Original Research 06 March 2017 Pages: 1117 - 1126
Synthesis and biological evaluation of 1,3,4-trisubstituted pyrazole analogues as anti-mycobacterial agents Shankar G. AlegaonMita B. HirparaV. M. Kumbar Original Research 06 March 2017 Pages: 1127 - 1138
Design, characterization, in vitro antibacterial, antitubercular evaluation and structure–activity relationships of new hydrazinyl thiazolyl coumarin derivatives Samina KhanYusufzaiHasnah OsmanNoviany Original Research 07 March 2017 Pages: 1139 - 1148
Synthesis, protease inhibition, and antileishmanial activity of new benzoxazoles derived from acetophenone or benzophenone and synthetic precursors Laís R. S. FolquittoPriscila F. NogueiraDanielle F. Dias Original Research 10 March 2017 Pages: 1149 - 1159
Novel iron phenanthroline-based photosensitizers for antimicrobial PDT: synthesis, DNA binding and photo-induced DNA cleavage activity Chittanahalli N. SudhamaniHalehatty S. Bhojya NaikPasupanetti N. Prashanth Kumar Original Research 11 March 2017 Pages: 1160 - 1169
In vitro production of reactive oxygen species (ROS) by sampangine Hamid R. NasiriKatharina HohmannHarald Schwalbe Original Research 12 March 2017 Pages: 1170 - 1175
N-alkylated thiazolidine-2,4-dione analogs as PTP1B inhibitors: synthesis, biological activity, and docking studies Manoj K. MahapatraRajnish KumarManoj Kumar Original Research 13 March 2017 Pages: 1176 - 1183
An improvement on the prediction power of the 3D-QSAR CoMFA models using a hybrid of statistical and machine learning methods: a case study on γ‑secretase modulators of Alzheimer’s disease Hadi KhaniMohammad B. SepehrifarShantia Yarahmadian Original Research 14 March 2017 Pages: 1184 - 1200
Novel quinoline bearing sulfonamide derivatives and their cytotoxic activity against MCF7 cell line N. S. AhmedK. O. BadahdahH. M. Qassar Original Research 14 March 2017 Pages: 1201 - 1212
Synthesis, spectral, biological activity, and crystal structure evaluation of novel pyrazoline derivatives having sulfonamide moiety Rajitha SadashivaDamodara NaralKudigana Jayaprakash Pampa Original Research 15 March 2017 Pages: 1213 - 1227
Design and synthesis of three series of novel antitumor–azo derivatives Phoebe F. LamieJohn N. Philoppes Original Research 15 March 2017 Pages: 1228 - 1240
Deoxypodophyllotoxin, a semi-synthetic compound from Dysosma versipellis, induces selective cell death in human breast cancer cell lines Meyada KhaledGhania BelaalouiLu-Yong Zhang Original Research 15 March 2017 Pages: 1241 - 1258
Atomic 3D-QSAR study based on pharmacophore modeling of resveratrol derivatives as selective COX-2 inhibitors Samira feddalZohra BouakoukSafia Kellou-Tairi Original Research 16 March 2017 Pages: 1259 - 1267
Bis-indole alkaloids from Tabernaemontana divaricata as potent pancreatic lipase inhibitors: molecular modelling studies and experimental validation Sridhar S. N. C.Seshank MutyaAtish T. Paul Original Research 16 March 2017 Pages: 1268 - 1278
Podophyllum derivatives containing fluorine atom in the 3-position of 2-aminopyridine improved the antitumor activity by inducing P53-dependent apoptosis Huai Wang Original Research 16 March 2017 Pages: 1279 - 1290
Potent cytotoxicity against human small cell lung cancer cells of the heptenes from the stem bark of Xylopia pierrei Hance Ratchanaporn ChokchaisiriSukanya KunkaewomApichart Suksamrarn Original Research 16 March 2017 Pages: 1291 - 1296
The influence of genistein on free radicals in normal dermal fibroblasts and keloid fibroblasts examined by EPR spectroscopy Magdalena JurzakPaweł RamosBarbara Pilawa Original Research Open access 16 March 2017 Pages: 1297 - 1305
Synthesis, docking, and evaluation of novel thiazoles for potent antidiabetic activity T. V. SravanthiS. Sajitha LuluS. L. Manju Original Research 16 March 2017 Pages: 1306 - 1315
Antibacterial properties of 5-substituted derivatives of rhodanine-3-carboxyalkyl acids Waldemar TejchmanIzabela Korona-GlowniakPiotr Suder Original Research Open access 16 March 2017 Pages: 1316 - 1324
A simple method for the synthesis of 1,3-diaminopropan-2-ols derivatives and their ex vivo relaxant activity on isolated rat tracheal rings Fabiola I. LópezFabiola N. de la CruzMiguel A. Vázquez Original Research 16 March 2017 Pages: 1325 - 1335
Ganoderic acid modulating TNF and its receptors: in silico and in vitro study Balraj Singh GillNavgeetSanjeev Kumar Original Research 16 March 2017 Pages: 1336 - 1348