Development of drugs based on imidazole and benzimidazole bioactive heterocycles: recent advances and future directions Monika GabaChander Mohan Review Article 31 December 2015 Pages: 173 - 210
Fluorine-containing benzothiazole as a novel trypanocidal agent: design, in silico study, synthesis and activity evaluation Roberto I. Cuevas-HernándezJosé Correa-BasurtoJosé G. Trujillo-Ferrara Original Research 15 October 2015 Pages: 211 - 224
Synthesis of 2-(2-methoxyphenyl)-5-phenyl-1,3,4-oxadiazole derivatives and evaluation of their antiglycation potential Muhammad TahaNor Hadiani IsmailMohd Zulkefeli Original Research 05 November 2015 Pages: 225 - 234
Synthesis, antimicrobial activities and QSAR studies of heterocyclic Schiff base ligands with organosilicon(IV) halides Jai DeviSuman KumariRajesh Malhotra Original Research 07 November 2015 Pages: 235 - 246
Synthesis and antimalarial activity of new nanocopolymer β-lactams and molecular docking study of their monomers Edris EbrahimiAliasghar JarrahpourEdward Turos Original Research 12 November 2015 Pages: 247 - 262
Design, synthesis and mode of action of novel 2-(4-aminophenyl)benzothiazole derivatives bearing semicarbazone and thiosemicarbazone moiety as potent antimicrobial agents Meenakshi SinghSudhir Kumar SinghSushil K. Singh Original Research 23 November 2015 Pages: 263 - 282
Novel 2-(1-(substitutedbenzyl)-1H-tetrazol-5-yl)-3-phenylacrylonitrile derivatives: synthesis, in vitro antitumor activity and computational studies Suresh MaddilaKovashnee NaickerSreekantha B. Jonnalagadda Original Research 30 November 2015 Pages: 283 - 291
Synthesis of some new thiazolo[3,2-a]pyrimidine derivatives and screening of their in vitro antibacterial and antitubercular activities Dong CaiZhi-Hua ZhangBing-Jie Fu Original Research 01 December 2015 Pages: 292 - 302
In vitro cytotoxicity study of ent-kaurenoic acid derivatives against human breast carcinoma cell line Marília R. SimãoLuiza J. CarneiroCassia S. Mizuno Original Research 06 December 2015 Pages: 303 - 309
Synthesis and CYP17α hydroxylase inhibition activity of new 3α- and 3β-ester derivatives of pregnenolone and related ether analogues Najim A. Al-MasoudiNabeel A. Abdul-RidaBahjat A. Saeed Original Research 08 December 2015 Pages: 310 - 321
Structure and toxicity of clozapine and olanzapine on agranulocytosis Rosivaldo S. BorgesGláucio R. NagurniakAlbérico B. F. da Silva Original Research 12 December 2015 Pages: 322 - 328
Synthesis and biological evaluation of 1,3,4-oxadiazole bearing dihydropyrimidines as potential antitubercular agents N. C. DesaiA. R. TrivediK. A. Bhatt Original Research 17 December 2015 Pages: 329 - 338
Synthesis, antimicrobial activity and docking studies of new N-ethyl-3-indolyl heterocycles Weal A. El-SayedHebat-Allah S. AbbasTomasz Magdziarz Original Research 23 December 2015 Pages: 339 - 355
Design, synthesis and neuraminidase inhibitory activity of N-(5-benzyl-4-(tert-butyl)thiazol-2-yl)benzamides Zhilin WuJunmei PengGuoxi Li Original Research 31 December 2015 Pages: 356 - 368
Synthesis and antimicrobial activity of some novel substituted pyridazin-3(2H)-ones containing 1,3,4-thiadiazole moiety Mohammed S. SallamMaher A. El-HashashDalal B. Guirguis Original Research 31 December 2015 Pages: 369 - 380