Guest Editorial Gianfabio GiorgioniAlessandro PiergentiliRichard A. Glennon EditorialNotes Pages: 1 - 4
The Nicotinic Acetylcholine Receptor: 25 Years Thereafter Ferdinand HuchoChristoph Weise OriginalPaper Pages: 11 - 17
Monitoring Receptor Dimerisation Graeme MilliganGeraldine PascalJuan J. Carrillo OriginalPaper Pages: 18 - 24
Heterodimerization of G-Protein-Coupled Receptors Reveals an Unexpected Level of Pharmacological Diversity Roberto MaggioMarco ScarselliGiovanni U. Corsini OriginalPaper Pages: 25 - 33
The Activation Mechanism of Class-III G-Protein Coupled Receptors J.-P. PinJ. KniazeffL. Prézeau OriginalPaper Pages: 38 - 51
Allosteric Regulation of Binding and Function at GCPRS Nigel J.M. BirdsallChristopher BrowningSebastian Lazareno OriginalPaper Pages: 52 - 62
Polyamines May Modulate Both G Protein-Coupled Receptors and G Proteins Gabriella MarucciFrancesca NoviCarlo Melchiorre OriginalPaper Pages: 63 - 73
Improgan-like Analgesics: A Family of Compounds Derived From Histamine Anatgonists L.B. HoughJ.W. NalwalkH. Timmerman OriginalPaper Pages: 78 - 87
Potent, Selective Adenosine A1 Agonists as Potential Analgesics P.J. BeswickC. BountraD.J. Spalding OriginalPaper Pages: 88 - 98
Introduction to Receptors in Aging Diseases: GABA Receptors Wolfgang Froestl OriginalPaper Pages: 99 - 102
Mechanisms and Issues Relating to the Use of D1-like Dopamine Receptor Agonists for Age-related Illnesses: Parkinson’s Disease and Memory and Cognition David E. NicholsMechelle M. Lewis OriginalPaper Pages: 105 - 114
Novel Mechanisms of Drug Action: Functional Selectivity at D2 Dopamine Receptors Richard B. MailmanElaine A. Gay OriginalPaper Pages: 115 - 126