1. Synthesis of new 7-chloro-4-phenoxyquinoline analogues as potential antitubercular agents

   • Preeti S. Salve
   • Shankar G. Alegaon

   Original Research 07 July 2017 Pages: 1 - 14

   

2. Synthesis, characterization and evaluation of cytotoxic and antioxidant activities of dihydropyrimidone substituted pyrrole derivatives

   • Asieh Khalilpour
   • Sakineh Asghari

   Original Research 28 August 2017 Pages: 15 - 22

   

3. Enriching biologically relevant chemical space around 2-aminothiazole template for anticancer drug development

   • Sarah Titus
   • Kumaran G. Sreejalekshmi

   Original Research 28 August 2017 Pages: 23 - 36

   

4. Isolation, purification and identification of antioxidants from Lepidium latifolium extracts

   • Yuan Xiang
   • Wang Haixia
   • Tao Yanduo

   Original Research 28 August 2017 Pages: 37 - 45

   

5. Antinociceptive property of vinyl sulfides in spite of their weak antioxidant activity

   • Francine R. Ianiski
   • Mariana M. Bassaco
   • Cristiane Luchese

   Original Research 28 August 2017 Pages: 46 - 51

   

6. Synthesis and antimicrobial activity of some heterocyclic compounds bearing benzimidazole and pyrazoline motifs

   • N. C. Desai
   • Darshan Pandya
   • Darshita Vaja

   Original Research 29 August 2017 Pages: 52 - 60

   

7. Synthesis and PASS-assisted evaluation of coumarin–benzimidazole derivatives as potential anti-inflammatory and anthelmintic agents

   • Purva Sethi
   • Yogita Bansal
   • Gulshan Bansal

   Original Research 29 August 2017 Pages: 61 - 71

   

8. Synthesis, structural characterization and anticancer evaluation of pyrazole derivatives

   • Mohamed S. A. El-Gaby
   • Mustafa M. Ghorab
   • Hala. M. Aly

   Original Research 04 September 2017 Pages: 72 - 79

   

9. Anti-proliferative, structure–activity relationship of pyridinylchalcones and chromanones

   • Cherupally Dayakar
   • Pathi Suman
   • Bhimapaka China Raju

   Original Research 04 September 2017 Pages: 80 - 94

   

10. Molecular modeling, pK _a and thermodynamic values of asthma drugs

    • Mobina Alimohammady
    • Mansour Jahangiri
    • Hasan Tahermansouri

    Original Research 04 September 2017 Pages: 95 - 114

    

11. Ent-kaurane diterpenoids from the pericarps of Datura metel L. acted on the vascular endothelial cells via TRPC6 and NF-κB protein

    • Bing-you Yang
    • Yong-qiang Zhou
    • Hai-xue Kuang

    Original Research 05 September 2017 Pages: 115 - 121

    

12. Relaxant effect of structurally related flavonoids on isolated tracheal rat rings: a SAR study

    • Angélica Flores-Flores
    • Sergio Hidalgo-Figueroa
    • Samuel Estrada-Soto

    Original Research 05 September 2017 Pages: 122 - 127

    

13. 3,5-Bis(2-fluorobenzylidene)-4-piperidone induce reactive oxygen species-mediated apoptosis in A549 cells

    • Guo-Yun Liu
    • Cong-Cong Jia
    • Jie Yang

    Original Research 05 September 2017 Pages: 128 - 136

    

14. Design, synthesis, characterization, and molecular modeling studies of novel oxadiazole derivatives of nipecotic acid as potential anticonvulsant and antidepressant agents

    • Ravi Bhushan Singh
    • Gireesh Kumar Singh
    • Md. Kamaruz Zaman

    Original Research 06 September 2017 Pages: 137 - 152

    

15. A novel chromonyl thiohydantoin with anti-proliferative action on primary hepatocellular carcinoma cells

    • Cigdem Ozen
    • Meltem Ceylan-Unlusoy
    • Oya Bozdag-Dundar

    Original Research 06 September 2017 Pages: 153 - 160

    

16. Synthesis, anti-lung cancer activity and molecular docking study of 3-methylene-2-oxoindoline-5-carboxamide derivatives

    • Juntao Ai
    • Meng Lv
    • Qianbin Li

    Original Research 06 September 2017 Pages: 161 - 170

    

17. One pot synthesis of thiazolo[2,3-b]dihydropyrimidinone possessing pyrazole moiety and evaluation of their anti-inflammatory and antimicrobial activities

    • Shivapura Viveka
    • Dinesha
    • Marikunte Yanjarappa Sreenivasa

    Original Research 07 September 2017 Pages: 171 - 185

    

18. The antinociceptive evaluation of 2,3-substituted-1,3-thiazolidin-4-ones through thermal stimulation in mice

    • Arthur H. S. Neves
    • Daniel S. da Silva
    • Adriana L. da Silva

    Original Research 08 September 2017 Pages: 186 - 193

    

19. Design, synthesis and anti-inflammatory activity of dihydroflavonol derivatives

    • Chunling Hu
    • Zongbao Zhou
    • Xiaochuan Ye

    Original Research 12 September 2017 Pages: 194 - 205

    

20. Design (Docking and QSAR Studies) and synthesis of histone deacetylase 2 (HDAC2) inhibitors series

    • Heidy Martínez-Pacheco
    • Judith Espinosa-Raya
    • Guillermo Ramírez-Galicia

    Original Research 12 September 2017 Pages: 206 - 223

    

21. Serendipitous formation of novel class of dichromeno pyrano pyrimidinone derivatives possessing anti-tubercular activity against M. tuberculosis H₃₇Rv

    • Nilam C. Dige
    • Prasad G. Mahajan
    • Dattaprasad M. Pore

    Original Research 12 September 2017 Pages: 224 - 233

    

22. Strategies to select the best pharmacophore model: a case study in pyrazoloquinazoline class of PLK-1 inhibitors

    • Akshada J. Joshi
    • Heena R. Bhojwani
    • Urmila J. Joshi

    Original Research 12 September 2017 Pages: 234 - 260

    

23. Vitamin K enhances the effect of antibiotics inhibiting the efflux pumps of Staphylococcus aureus strains

    • Saulo R. Tintino
    • Cícera D. M. Oliveira-Tintino
    • Valdir Q. Balbino

    Original Research 14 September 2017 Pages: 261 - 267

    

24. Triterpenoids from the stem bark of Vitellaria paradoxa (Sapotaceae) and derived esters exhibit cytotoxicity against a breast cancer cell line

    • Kenneth O. Eyong
    • Guerisson Bairy
    • Daniel Romo

    Original Research 14 September 2017 Pages: 268 - 277

    

25. Activity of ring-substituted 8-hydroxyquinoline-2-carboxanilides against intestinal sulfate-reducing bacteria Desulfovibrio piger

    • Ivan Kushkevych
    • Jiri Kos
    • Josef Jampilek

    Original Research 15 September 2017 Pages: 278 - 284

    

26. Design, synthesis, and cytotoxicity evaluation of threonine-based galactoceramide with aromatic groups and various fatty-acyl side chains

    • Srikanth Vudhgiri
    • Sunitha Rani Routhu
    • Ram Chandra Reddy Jala

    Original Research 15 September 2017 Pages: 285 - 307

    

27. Evaluation of heteroatom-rich derivatives as antitubercular agents with InhA inhibition properties

    • Bachar Rébat Moulkrere
    • Beatrice S. Orena
    • Mokhtar Fodili

    Original Research 15 September 2017 Pages: 308 - 320

    

28. Novel indole derivatives as potential anticancer agents: Design, synthesis and biological screening

    • B. Prakash
    • A. Amuthavalli
    • R. Velmurugan

    Original Research 18 September 2017 Pages: 321 - 331

    

29. Molecular docking, binding free energy analysis, and biological evaluation of bisabolonalone hydrazone carboxamides as H⁺,K⁺-ATPase reversible inhibitors

    • Xin-Xin She
    • Qing Dong
    • Kun Zou

    Original Research 18 September 2017 Pages: 332 - 340

    

30. Integrated in silico–in vitro screening of ovarian cancer peroxisome proliferator-activated receptor-γ agonists against a biogenic compound library

    • Gui-Lian Zhang
    • Feng-Ying Liu
    • Shi-Ming Lv

    Original Research 19 September 2017 Pages: 341 - 349