Volume 9, issue 1, December 2024
45 articles in this issue
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eTFC-01: a dual-labeled chelate-bridged tracer for SSTR2-positive tumors
Authors (first, second and last of 7)
- Dylan Chapeau
- Savanne Beekman
- Yann Seimbille
- Content type: Research article
- Open Access
- Published: 22 May 2024
- Article: 44
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In vitro and in vivo evaluation of a tetrazine-conjugated poly-L-lysine effector molecule labeled with astatine-211
Authors (first, second and last of 6)
- Chiara Timperanza
- Holger Jensen
- Emma Aneheim
- Content type: Research article
- Open Access
- Published: 22 May 2024
- Article: 43
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Highlight selection of radiochemistry and radiopharmacy developments by editorial board
Authors (first, second and last of 24)
- Jun Toyohara
- Danielle Vugts
- Cécile Bourdeau
- Content type: Review
- Open Access
- Published: 16 May 2024
- Article: 42
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[68Ga]Ga-NODAGA-TriGalactan, a low molecular weight tracer for the non-invasive imaging of the functional liver reserve
Authors (first, second and last of 9)
- Maximilian A. Zierke
- Christine Rangger
- Roland Haubner
- Content type: Research article
- Open Access
- Published: 15 May 2024
- Article: 41
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Good practices for 89Zr radiopharmaceutical production and quality control
Authors (first, second and last of 4)
- Thomas Erik Wuensche
- Serge Lyashchenko
- Danielle Vugts
- Content type: Review
- Open Access
- Published: 11 May 2024
- Article: 40
This is part of 1 collection: -
Automated synthesis of [89Zr]ZrCl4, [89Zr]ZrDFOSquaramide-bisPh(PSMA) and [89Zr]ZrDFOSquaramide-TATE
Authors (first, second and last of 6)
- Asif Noor
- Peter D. Roselt
- Paul S. Donnelly
- Content type: Research article
- Open Access
- Published: 08 May 2024
- Article: 39
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Bifunctional octadentate pseudopeptides as Zirconium-89 chelators for immuno-PET applications
Authors (first, second and last of 12)
- Valentina Albanese
- Chiara Roccatello
- Emiliano Cazzola
- Content type: Research article
- Open Access
- Published: 06 May 2024
- Article: 38
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Radiation nanomedicines for cancer treatment: a scientific journey and view of the landscape
Authors (first, second and last of 4)
- Raymond M. Reilly
- Constantine J. Georgiou
- Zhongli Cai
- Content type: Review
- Open Access
- Published: 04 May 2024
- Article: 37
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99mTc-labeled FAPI compounds for cancer and inflammation: from radiochemistry to the first clinical applications
Authors (first, second and last of 5)
- Alessandra Boschi
- Luca Urso
- Luca Filippi
- Content type: Review
- Open Access
- Published: 02 May 2024
- Article: 36
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GMP production of [18F]FE-PE2I on a TRACERLab FX2 N synthesis module, a radiotracer for in vivo PET imaging of the dopamine transport
Authors (first, second and last of 11)
- Mélodie Ferrat
- Mohammad M. Moein
- Thuy A. Tran
- Content type: Methodology
- Open Access
- Published: 02 May 2024
- Article: 35
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Advancing 6-bromo-7-[11C]methylpurine to clinical use: improved regioselective radiosynthesis, non-clinical toxicity data and human dosimetry estimates
Authors (first, second and last of 10)
- Severin Mairinger
- Matthias Jackwerth
- Oliver Langer
- Content type: Research article
- Open Access
- Published: 29 April 2024
- Article: 34
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Small animal PET imaging with the 68Ga-labeled pH (low) insertion peptide-like peptide YJL-4 in a triple-negative breast cancer mouse model
Authors (first, second and last of 7)
- YueHua Chen
- ShuangShuang Song
- MingMing Yu
- Content type: Research article
- Open Access
- Published: 27 April 2024
- Article: 33
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Radiolabeled 15-mer peptide internalization is mediated by megalin (LRP2 receptor) in a CRISPR/Cas9-based LRP2 knockout human kidney cell model
Authors (first, second and last of 8)
- Anna Durinova
- Lucie Smutna
- Frantisek Trejtnar
- Content type: Research article
- Open Access
- Published: 18 April 2024
- Article: 32
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Automated radiolabelling of [68Ga]Ga-PSMA-11 (gallium (68Ga)-gozetotide) using the Locametz® kit and two generators
Authors (first, second and last of 5)
- Elke A. van Brandwijk
- Else A. Aalbersberg
- Jeroen J. M. A. Hendrikx
- Content type: Research article
- Open Access
- Published: 17 April 2024
- Article: 31
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Comparison of approaches for increasing affinity of affibody molecules for imaging of B7-H3: dimerization and affinity maturation
Authors (first, second and last of 6)
- Maryam Oroujeni
- Matilda Carlqvist
- Fredrik Y. Frejd
- Content type: Research article
- Open Access
- Published: 16 April 2024
- Article: 30
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Production of [211At]NaAt solution under GMP compliance for investigator-initiated clinical trial
Authors (first, second and last of 12)
- Sadahiro Naka
- Kazuhiro Ooe
- Tadashi Watabe
- Content type: Research article
- Open Access
- Published: 15 April 2024
- Article: 29
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Improved automated one-pot two-step radiosynthesis of (S)-[18F]FETrp, a radiotracer for PET imaging of indoleamine 2,3-dioxygenase 1 (IDO1)
Authors (first, second and last of 7)
- Aurélie Maisonial-Besset
- David Kryza
- Jean-Michel Chezal
- Content type: Research article
- Open Access
- Published: 02 April 2024
- Article: 28
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Human biodistribution and radiation dosimetry for the tau tracer [18F]Florzolotau in healthy subjects
Authors (first, second and last of 5)
- Kun-Ju Lin
- Shao-Yi Huang
- Ing-Tsung Hsiao
- Content type: Research article
- Open Access
- Published: 02 April 2024
- Article: 27
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In vivo evaluation of tumor uptake and bio-distribution of 99mTc-labeled 1-thio-β-D-glucose and 5-thio-D-glucose in mice model
Authors (first, second and last of 13)
- Fabian Muehlberg
- Konrad Mohnike
- Max Seidensticker
- Content type: Research article
- Open Access
- Published: 29 March 2024
- Article: 26
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Expanding a peptide-covalent probe hybrid for PET imaging of S. aureus driven focal infections
Authors (first, second and last of 8)
- Jyotsna Bhatt Mitra
- Saurav Chatterjee
- Archana Mukherjee
- Content type: Research article
- Open Access
- Published: 26 March 2024
- Article: 25
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In-target production of [11C]CH4 from a nitrogen/hydrogen gas target as a function of beam current, irradiation time, and target temperature
Authors (first, second and last of 6)
- Semi Helin
- Johan Rajander
- Olof Solin
- Content type: Research article
- Open Access
- Published: 25 March 2024
- Article: 24
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Validation of a size exclusion method for concomitant purification and formulation of peptide radiopharmaceuticals
Authors (first, second and last of 5)
- Sebastian Martin
- Lennard Wendlinger
- Margret Schottelius
- Content type: Methodology
- Open Access
- Published: 21 March 2024
- Article: 23
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Correction: Physiologically based radiopharmacokinetic (PBRPK) modeling to simulate and analyze radiopharmaceutical therapies: studies of non-linearities, multi-bolus injections, and albumin binding
Authors (first, second and last of 4)
- Ali Fele‑Paranj
- Babak Saboury
- Arman Rahmim
- Content type: Correction
- Open Access
- Published: 19 March 2024
- Article: 22
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Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
Authors (first, second and last of 9)
- Eva Schlein
- Johanna Rokka
- Jonas Eriksson
- Content type: Research article
- Open Access
- Published: 06 March 2024
- Article: 21
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Preclinical characterisation of gallium-68 labeled ferrichrome siderophore stereoisomers for PET imaging applications
Authors (first, second and last of 7)
- Kristyna Krasulova
- Barbora Neuzilova
- Milos Petrik
- Content type: Research article
- Open Access
- Published: 04 March 2024
- Article: 20
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A novel PET probe to selectively image heat shock protein 90α/β isoforms in the brain
Authors (first, second and last of 15)
- Takayuki Sakai
- Aya Ogata
- Yasuyuki Kimura
- Content type: Research article
- Open Access
- Published: 04 March 2024
- Article: 19
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Preclinical comparison of [177Lu]Lu-rhPSMA-10.1 and [177Lu]Lu-rhPSMA-10.2 for endoradiotherapy of prostate cancer: biodistribution and dosimetry studies
Authors (first, second and last of 9)
- Alexander Wurzer
- Francesco De Rose
- Calogero D’Alessandria
- Content type: Research article
- Open Access
- Published: 26 February 2024
- Article: 18
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Neopentyl glycol-based radiohalogen-labeled amino acid derivatives for cancer radiotheranostics
Authors (first, second and last of 12)
- Yuta Kaizuka
- Hiroyuki Suzuki
- Tomoya Uehara
- Content type: Research article
- Open Access
- Published: 26 February 2024
- Article: 17
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Radiosynthesis, structural identification and in vitro tissue binding study of [18F]FNA-S-ACooP, a novel radiopeptide for targeted PET imaging of fatty acid binding protein 3
Authors (first, second and last of 11)
- Pyry Dillemuth
- Tuomas Karskela
- Xiang-Guo Li
- Content type: Research article
- Open Access
- Published: 23 February 2024
- Article: 16
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Optimization and scale up of production of the PSMA imaging agent [18F]AlF-P16-093 on a custom automated radiosynthesis platform
Authors (first, second and last of 7)
- David Alexoff
- Seok Rye Choi
- Hank Kung
- Content type: Research article
- Open Access
- Published: 23 February 2024
- Article: 15
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Chelator impact: investigating the pharmacokinetic behavior of copper-64 labeled PD-L1 radioligands
Authors
- Fabian Krutzek
- Cornelius K. Donat
- Sven Stadlbauer
- Content type: Research article
- Open Access
- Published: 19 February 2024
- Article: 14
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Preclinical evaluation of new GRPR-antagonists with improved metabolic stability for radiotheranostic use in oncology
Authors (first, second and last of 8)
- Panagiotis Kanellopoulos
- Adam Mattsson
- Anna Orlova
- Content type: Research article
- Open Access
- Published: 16 February 2024
- Article: 13
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Intranasal administration enhances size-dependent pulmonary phagocytic uptake of poly(lactic-co-glycolic acid) nanoparticles
Authors (first, second and last of 7)
- Seung Ho Baek
- Eun-Ha Hwang
- Jung Joo Hong
- Content type: Research article
- Open Access
- Published: 15 February 2024
- Article: 12
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Validation of an automated dispensing system for subsequent dose dispensing of different radionuclides
Authors (first, second and last of 4)
- T. T. Cao
- E. A. Aalbersberg
- J. J. M. A. Hendrikx
- Content type: Research article
- Open Access
- Published: 12 February 2024
- Article: 11
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Improved synthesis of 6-bromo-7-[11C]methylpurine for clinical use
Authors (first, second and last of 4)
- Toshimitsu Okamura
- Tatsuya Kikuchi
- Ming-Rong Zhang
- Content type: Research article
- Open Access
- Published: 09 February 2024
- Article: 10
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Implementing Ac-225 labelled radiopharmaceuticals: practical considerations and (pre-)clinical perspectives
Authors (first, second and last of 7)
- Eline L. Hooijman
- Valery Radchenko
- Erik de Blois
- Content type: Review
- Open Access
- Published: 06 February 2024
- Article: 9
This is part of 1 collection: -
Unnatural amino acid substitutions to improve in vivo stability and tumor uptake of 68Ga-labeled GRPR-targeted TacBOMB2 derivatives for cancer imaging with positron emission tomography
Authors (first, second and last of 10)
- Lei Wang
- Hsiou-Ting Kuo
- Kuo-Shyan Lin
- Content type: Research article
- Open Access
- Published: 02 February 2024
- Article: 8
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A novel PSMA-targeting tracer with highly negatively charged linker demonstrates decreased salivary gland uptake in mice compared to [68Ga]Ga-PSMA-11
Authors (first, second and last of 4)
- Steve S. Huang
- Frank P. DiFilippo
- Warren D. Heston
- Content type: Research article
- Open Access
- Published: 30 January 2024
- Article: 7
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Physiologically based radiopharmacokinetic (PBRPK) modeling to simulate and analyze radiopharmaceutical therapies: studies of non-linearities, multi-bolus injections, and albumin binding
Authors (first, second and last of 4)
- Ali Fele-Paranj
- Babak Saboury
- Arman Rahmim
- Content type: Research article
- Open Access
- Published: 22 January 2024
- Article: 6
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Preclinical evaluation of the theranostic potential of 89Zr/177Lu-labeled anti-TROP-2 antibody in triple-negative breast cancer model
Authors (first, second and last of 6)
- Yitian Wu
- Tuo li
- Li Huo
- Content type: Research article
- Open Access
- Published: 09 January 2024
- Article: 5
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Cu(II)-Mediated direct 18F-dehydrofluorination of phosphine oxides in high molar activity
Authors (first, second and last of 5)
- Xiaoqun Tang
- Shengji Lv
- Zijing Li
- Content type: Methodology
- Open Access
- Published: 06 January 2024
- Article: 4
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Production of the PET radionuclide 61Cu via the 62Ni(p,2n)61Cu nuclear reaction
Authors (first, second and last of 4)
- Santiago Andrés Brühlmann
- Martin Walther
- Martin Kreller
- Content type: Research article
- Open Access
- Published: 05 January 2024
- Article: 3
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Position paper to facilitate patient access to radiopharmaceuticals: considerations for a suitable pharmaceutical regulatory framework
Authors (first, second and last of 15)
- Aruna Korde
- Marianne Patt
- Clemens Decristoforo
- Content type: Position paper
- Open Access
- Published: 02 January 2024
- Article: 2
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Preclinical evaluation of an 18F-labeled Nε-acryloyllysine piperazide for covalent targeting of transglutaminase 2
Authors (first, second and last of 9)
- Robert Wodtke
- Markus Laube
- Reik Löser
- Content type: Research article
- Open Access
- Published: 02 January 2024
- Article: 1