Expression of Multidrug Resistance-Associated Protein (MRP) in Human Retinal Pigment Epithelial Cells and Its Interaction with BAPSG, a Novel Aldose Reductase Inhibitor Jithan V. AukunuruGangadhar SunkaraUday B. Kompella OriginalPaper Pages: 565 - 572
Transport of Levofloxacin in the OK Kidney Epithelial Cell Line: Interaction with p-Aminohippurate Transport Yumiko MatsuoIkuko YanoKen–ichi Inui OriginalPaper Pages: 573 - 578
Physicochemical Parameters Responsible for the Affinity of Methotrexate Analogs for Rat Canalicular Multispecific Organic Anion Transporter (cMOAT/MRP2) Yong–Hae HanYukio KatoYuichi Sugiyama OriginalPaper Pages: 579 - 586
P-Glycoprotein Inhibition Leads to Enhanced Disruptive Effects by Anti-Microtubule Cytostatics at the In Vitro Blood-Brain Barrier Inez C. J. van der SandtPieter J. GaillardDouwe D. Breimer OriginalPaper Pages: 587 - 592
Influence of a Microemulsion Vehicle on Cutaneous Bioequivalence of a Lipophilic Model Drug Assessed by Microdialysis and Pharmacodynamics Mads KreilgaardMichiel J. B. KemmeAdam F. Cohen OriginalPaper Pages: 593 - 599
Synthesis, In Vitro Skin Permeation Studies, and PLS-Analysis of New Naproxen Derivatives Horst WeberUta SteimerGabriele Cruciani OriginalPaper Pages: 600 - 607
Mutual Inhibition of the Insulin Absorption-Enhancing Properties of Dodecylmaltoside and Dimethyl-β-cyclodextrin Following Nasal Administration Fakhrul AhsanJohn J. ArnoldDennis J. Pillion OriginalPaper Pages: 608 - 614
CYP2C19 Genotype Related Effect of Omeprazole on Intragastric pH and Antimicrobial Stability Tomoko KitaYusuke TanigawaraMasato Kasuga OriginalPaper Pages: 615 - 621
Inhibition of In Vitro Metabolism of Simvastatin by Itraconazole in Humans and Prediction of In Vivo Drug-Drug Interactions Michi IshigamMinoru UchiyamaYuichi Sugiyama OriginalPaper Pages: 622 - 631
Effect of Oxidative Stress on the Structure and Function of Human Serum Albumin Makoto AnrakuKeishi YamasakiMasaki Otagiri OriginalPaper Pages: 632 - 639
Development of Systems for Targeting the Regional Lymph Nodes for Diagnostic Imaging: In Vivo Behaviour of Colloidal PEG-Coated Magnetite Nanospheres in the Rat Following Interstitial Administration L. IllumA. E. ChurchS. S. Davis OriginalPaper Pages: 640 - 645
Relationship Between Physicochemical and Osteotropic Properties of Bisphosphonic Derivatives: Rational Design for Osteotropic Drug Delivery System (ODDS) Hideki HirabayashiTaiji SawamotoTakehisa Hata OriginalPaper Pages: 646 - 651
Development of a Generalized, Quantitative Physicochemical Model of CYP3A4 Inhibition for Use in Early Drug Discovery R. J. RileyA. J. ParkerC. N. Manners OriginalPaper Pages: 652 - 655
SEM Imaging Predicts Quality of Niosomes from Maltodextrin-Based Proniosomes Almira I. Blazek–WelshDavid G. Rhodes OriginalPaper Pages: 656 - 661
The Use of Inverse Phase Gas Chromatography to Measure the Surface Energy of Crystalline, Amorphous, and Recently Milled Lactose Helen E. NewellGraham BucktonDaryl R. Williams OriginalPaper Pages: 662 - 666
Effect of Cyclodextrin Charge on Complexation of Neutral and Charged Substrates: Comparison of (SBE)7M-β-CD to HP-β-CD V. ZiaR. A. RajewskiV. J. Stella OriginalPaper Pages: 667 - 673
Microhardness and Dislocation Identification Studies on Paracetamol Single Crystals Stuart FinnieKorlakunte V. R. PrasadJohn N. Sherwood OriginalPaper Pages: 674 - 681
Polymorph Control of Sulfathiazole in Supercritical CO2 A. KordikowskiT. ShekunovP. York OriginalPaper Pages: 682 - 688
Study of the Breakup Under Shear of a New Thermally Reversible Water-in-Oil-in-Water (W/O/W) Multiple Emulsion Laetitia OlivieriMonique SeillerJean–Louis Grossiord OriginalPaper Pages: 689 - 693
Lipophilicity Behaviour of the Zwitterionic Antihistamine Cetirizine in Phosphatidylcholine Liposomes/Water Systems Georgette Plemper van BalenGiulia CaronBernard Testa OriginalPaper Pages: 694 - 701
The Apparent Lipophilicity of Quaternary Ammonium Ions Is Influenced by Galvani Potential Difference, Not Ion-Pairing: A Cyclic Voltammetry Study Géraldine BouchardPierre–Alain CarruptHubert H. Girault OriginalPaper Pages: 702 - 708
The Preparation, Characterization, and Evaluation of Cationic Microparticles for DNA Vaccine Delivery M. BrionesM. SinghD. O'Hagan OriginalPaper Pages: 709 - 712
Effects of Tacrolimus and Cyclosporin A on Peptide Transporter PEPT1 in Caco-2 Cells Hideyuki MotohashiToshiya KatsuraKen-ichi Inui OriginalPaper Pages: 713 - 717