Behavior of Hygroscopic Pharmaceutical Aerosols and the Influence of Hydrophobic Additives Anthony J. HickeyTed B. Martonen ReviewPaper Pages: 1 - 7
Mean Residence Time of Oral Drugs Undergoing First-Pass and Linear Reversible Metabolism Haiyung ChengWilliam J. Jusko OriginalPaper Pages: 8 - 13
Enantioselective Pharmacokinetics of dl-threo-Methylphenidate in Humans Nuggehally R. SrinivasJohn W. HubbardKamal K. Midha OriginalPaper Pages: 14 - 21
Pharmacokinetics of Stereomeric 1,4:3,6-Dianhydrohexitol Mononitrates in Rats Tsang-Bin TzengHo-Leung Fung OriginalPaper Pages: 22 - 27
Steady-State Bioavailability and Day-to-Day Variability of a Multiple-Unit (CR/ZOK) and a Single-Unit (OROS) Delivery System of Metoprolol After Once-Daily Dosing Anders SandbergBertil AbrahamssonRobert Bergstrand OriginalPaper Pages: 28 - 34
Time-Dependent Disposition of β-Naphthoflavone in the Rat Adedayo AdedoyinLeon AaronsJ. Brian Houston OriginalPaper Pages: 35 - 43
Distribution of Tacrine Across the Blood–Brain Barrier in Awake, Freely Moving Rats Using in Vivo Microdialysis Sampling Martin Telting-DiazCraig E. Lunte OriginalPaper Pages: 44 - 48
Prinomide Tromethamine Pharmacokinetics: Mutually Dependent Saturable and Competitive Protein Binding Between Prinomide and Its Own Metabolite Gregory M. KochakSudhakar PaiHanspeter Egger OriginalPaper Pages: 49 - 55
Column-Switching High-Performance Liquid Chromatographic Determination of a 2-Pyridinone-Based Human Immunodeficiency Virus Type 1 (HlV-l)-Specific Reverse Transcriptase Inhibitor in Human Plasma Eric J. WoolfBogdan K. Matuszewski OriginalPaper Pages: 56 - 60
Changes in Material Properties Accompanying the National Formulary (NF) Identity Test for Microcrystalline Cellulose Harry G. BrittainGeoffrey LewenSusan Bogdanowich OriginalPaper Pages: 61 - 67
Prodrugs of Peptides. 18. Synthesis and Evaluation of Various Esters of Desmopressin (dDAVP) Anne H. KahnsAnders BuurHans Bundgaard OriginalPaper Pages: 68 - 74
The 3′-Keto–Diol Equilibrium of Trospectomycin Sulfate Bulk Drug and Freeze-Dried Formulation: Solid-State Carbon-13 Cross-Polarization Magic Angle Spinning (CP/MAS) and High-Resolution Carbon-13 Nuclear Magnetic Resonance (NMR) Spectroscopy Studies Michael D. LikarRichard J. TaylorRussell H. Robins OriginalPaper Pages: 75 - 79
Design of New Formulations for Topical Ocular Administration: Polymeric Nanocapsules Containing Metipranolol Cándida LosaLaurent Marchal-HeusslerMaria J. Alonso OriginalPaper Pages: 80 - 87
Compression Characteristics of Granulated Materials. VII. The Effect of Intragranular Binder Distribution on the Compactibility of Some Lactose Granulations Martin WikbergGöran Alderborn OriginalPaper Pages: 88 - 94
Chemical Pathways of Peptide Degradation. IV. Pathways, Kinetics, and Mechanism of Degradation of an Aspartyl Residue in a Model Hexapeptide Cecilia OliyaiRonald T. Borchardt OriginalPaper Pages: 95 - 102
Stability of β-Galactosidase, a Model Protein Drug, Is Related to Water Mobility as Measured by 17O Nuclear Magnetic Resonance (NMR) Sumie YoshiokaYukio AsoTadao Terao OriginalPaper Pages: 103 - 108
Controlled Delivery of Pilocarpine. 1. In Vitro Characterization of Gelfoam® Matrices Sreekant R. NadkarniSamuel H. Yalkowsky OriginalPaper Pages: 109 - 112
Comparison of the Permeability Characteristics of a Human Colonic Epithelial (Caco-2) Cell Line to Colon of Rabbit, Monkey, and Dog Intestine and Human Drug Absorption Werner RubasNancy JezykGeorge M. Grass OriginalPaper Pages: 113 - 118
Sustained Bronchodilation with Isoproterenol Poly(Glycolide-co-Lactide) Microspheres Yih-Loong LaiRahul C. MehtaPatrick P. DeLuca OriginalPaper Pages: 119 - 125
Human Transbuccal Absorption of Diclofenac Sodium from a Prototype Hydrogel Delivery Device James CassidyBret BernerMalcolm Rowland OriginalPaper Pages: 126 - 129
Regional Gastrointestinal Absorption of the Beta-Blocker Pafenolol in the Rat and Intestinal Transit Rate Determined by Movement of 14C-Polyethylene Glycol (PEG) 4000 Hans LennernäsCarl-Gunnar Regårdh OriginalPaper Pages: 130 - 135
Relationship Among Physicochemical Properties, Skin Permeability, and Topical Activity of the Racemic Compound and Pure Enantiomers of a New Antifungal Lorraine WearleyBarry AntonacciTaisa Yarosh-Tomaine OriginalPaper Pages: 136 - 140
Acacia-Gelatin Microencapsulated Liposomes: Preparation, Stability, and Release of Acetylsalicylic Acid Cunji DongJames A. Rogers OriginalPaper Pages: 141 - 146
Comparison of the Leakage of Carboxyfluorescein from Symmetric-and Asymmetric-Acyl Chain Phosphatidylcholine Vesicles Timothy S. WiedmannAmir SalmonWalter R. Perkins Note Pages: 147 - 151
Effect of Humidity and Occlusion on the Percutaneous Absorption of Parathion in Vitro Shao-Kaung ChangJim E. Riviere Note Pages: 152 - 155
Kinetics of Aspirin Hydrolysis and Stabilization in the Presence of 2-Hydroxypropyl-β-Cyclodextrin Somesh ChoudhuryAshim K. Mitra Note Pages: 156 - 159