Iodine-mediated \({ sp}^{3}\) C–H functionalization of methyl ketones: a one-pot synthesis of functionalized indolizines via the 1,3-dipolar cycloaddition reaction between pyridinium ylides and ynones Issa YavariJamil SheykhahmadiMohammad Reza Halvagar Original Article 11 January 2017 Pages: 1 - 8
Substituted tetrazoles as multipurpose screening compounds Nicole RügerGeorg Michael FassauerAndreas Link Original Article 27 December 2016 Pages: 9 - 27
Efficient one-pot synthesis of new 1-amino substituted pyrrolo[1,2-a]quinoline-4-carboxylate esters via copper-free Sonogashira coupling reactions Ali KeivanlooShaghayegh Sadat KazemiAbdolhamid Bamoniri Original Article 06 September 2016 Pages: 29 - 36
Synthesis of first ever 4-quinolone-3-carboxylic acid-appended spirooxindole-pyrrolidine derivatives and their biological applications Thangaraj ArasakumarSadasivam MathusaliniPalathurai Subramaniam Mohan Original Article 26 September 2016 Pages: 37 - 52
Novel benzothiophene 1,1-dioxide deoxygenation path for the microwave-assisted synthesis of substituted benzothiophene-fused pyrrole derivatives Hamza KarakuşYaşar Dürüst Original Article 27 September 2016 Pages: 53 - 60
Expanding indole diversity: direct 1-step synthesis of 1,2-fused indoles and spiroindolines from 2-halo anilines for fast SAR antiviral elucidation against tobacco mosaic virus (TMV) Linwei ChenYongxian LiuQingmin Wang Original Article 03 September 2016 Pages: 61 - 68
One-pot synthesis of \(\upgamma \)-spiroiminolactones and \(\upgamma \)-dispiroiminolactones using \(\textit{N}{,}{} \textit{N}^{\prime }\)-disubstituted parabanic acid and thioparabanic acid derivatives Sakineh AsghariMohammad QandaleeAmir Ali Sarmadi Original Article 20 September 2016 Pages: 69 - 79
Indium triflate promoted one-pot multicomponent synthesis of structurally diverse 3-amino-imidazo[1,2-a]pyridines Suman SwamiArunava AgarwalaRahul Shrivastava Original Article 26 September 2016 Pages: 81 - 88
Synthesis of amino ester-embedded benzimidazoles: a one-pot sequential protocol under metal-free neutral conditions Priyabrata RoyChandan BodhakAnimesh Pramanik Original Article 27 September 2016 Pages: 89 - 100
A versatile strategy for the design and synthesis of novel ADP conjugates and their evaluation as potential poly(ADP-ribose) polymerase 1 inhibitors Yuliya V. SherstyukAlexandra L. ZakharenkoTatyana V. Abramova Original Article 27 September 2016 Pages: 101 - 113
Synthesis and antibacterial evaluation of new N- and S-glycosides analogues with dinitrophenyl-substituted heterocyclic bases Fatima BelkhademAdil A. Othman Original Article 19 October 2016 Pages: 115 - 124
Synthesis and biological evaluation of N-(3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-7-yl)benzenesulfonamide derivatives as new BET bromodomain inhibitors for anti-hematologic malignancies activities Li LiuYongxia ZhuLuoting Yu Original Article 17 November 2016 Pages: 125 - 136
Synthesis and antimicrobial evaluation of ester-linked 1,4-disubstituted 1,2,3-triazoles with a furyl/thienyl moiety C. P. KaushikRaj LuxmiAshwani Kumar Original Article 29 November 2016 Pages: 137 - 145
A green one-pot three-component cascade reaction: the synthesis of 2-amino-5,8-dihydro-3H-pyrido[2,3-D]pyrimidin-4-ones in aqueous medium Ahmad ShaabaniHeshmatollah SepahvandMohammad Tayeb Faroghi Original Article 12 January 2017 Pages: 147 - 153
Functionalized ionic liquid-assisted chromatography-free synthesis of bis(indolyl)methanes Sunita ChoudharyKhima PandeyAnil Kumar Original Article 11 January 2017 Pages: 155 - 162
Design, synthesis, in silico and biological evaluation of novel 2-(4-(4-substituted piperazin-1-yl)benzylidene)hydrazine carboxamides Shikha KumariChandra Bhushan MishraManisha Tiwari Original Article 30 December 2016 Pages: 163 - 174
Identification of potential glutaminyl cyclase inhibitors from lead-like libraries by in silico and in vitro fragment-based screening Mária SzaszkóIstván HajdúGyörgy Dormán Original Article 09 January 2017 Pages: 175 - 186
Discovery of potent NEK2 inhibitors as potential anticancer agents using structure-based exploration of NEK2 pharmacophoric space coupled with QSAR analyses Mohammad A. KhanfarFahmy BanatSaja Alqtaishat Original Article 06 September 2016 Pages: 187 - 200
Antioxidative and antiproliferative activities of novel pyrido[1,2-a]benzimidazoles Martina TireliKristina StarčevićMarijana Hranjec Original Article 27 September 2016 Pages: 201 - 210
QSAR models of antiproliferative activity of imidazo[2,1-b][1,3,4]thiadiazoles in various cancer cell lines Joanna MatysiakAndrzej Niewiadomy Original Article 08 October 2016 Pages: 211 - 218
Molecular topology: a strategy to identify novel compounds against ulcerative colitis María Gálvez-LlompartMaria C. RecioJorge Gálvez ORIGINAL ARTICLE 12 October 2016 Pages: 219 - 234
Computer modeling in predicting the bioactivity of human 5-lipoxygenase inhibitors Mengdi ZhangZhonghua XiaAixia Yan Original Article 30 November 2016 Pages: 235 - 246
A facile, efficient, and sustainable chitosan/CaHAp catalyst and one-pot synthesis of novel 2,6-diamino-pyran-3,5-dicarbonitriles Suresh MaddilaKranthi Kumar GanguSreekantha B. Jonnalagadda Short Communication 17 November 2016 Pages: 247 - 255
