Ring-closing metathesis as key step in the synthesis of Luffarin I, 16-epi-Luffarin I and Luffarin A Aitor UrosaIsidro S. MarcosPilar Basabe Full-Length Paper 20 October 2015 Pages: 369 - 377
A facile, regioselective synthesis of novel 3-(N-phenylcarboxamide)pyrazolo[1,5-a]pyrimidine analogs in the presence of KHSO\(_{4}\) in aqueous media assisted by ultrasound and their antibacterial activities Shunan KapingIvee BoissJai N. Vishwakarma Full-Length Paper 28 October 2015 Pages: 379 - 390
Synthesis and antimicrobial evaluation of novel 4-amino-6-(1,3,4-oxadiazolo/1,3,4-thiadiazolo)-pyrimidine derivatives Poornima ShettyB. M. PraveenSrinivas Cheruku Full-Length Paper 26 October 2015 Pages: 391 - 398
Synthesis and antitumor evaluation of novel sulfonylcycloureas derived from nitrogen mustard H. CheloufiB. BelhaniM. Berredjem Full-Length Paper 23 November 2015 Pages: 399 - 405
Tuning the Lewis acid phenol \(\varvec{ortho}\)-prenylation as a molecular diversity tool Sebastián N. JägerExequiel O. J. PortaGuillermo R. Labadie Full-Length Paper 03 November 2015 Pages: 407 - 419
Integrating sampling techniques and inverse virtual screening: toward the discovery of artificial peptide-based receptors for ligands Germán M. PérezLuis A. SalomónMarcello Mascini Full-Length Paper 09 November 2015 Pages: 421 - 438
Discovery of Influenza A virus neuraminidase inhibitors using support vector machine and Naïve Bayesian models Wenwen LianJiansong FangGuan-Hua Du Full-Length Paper 21 December 2015 Pages: 439 - 451
Combinatorial synthesis of deuterium-enriched atorvastatin Feng LiWenfeng JiangWenbao Li Original Article 25 January 2016 Pages: 453 - 459
A novel four- and pseudo-five-component reaction: unexpected efficient one-pot synthesis of 4H-thiopyran derivatives Akbar MobinikhalediMohammad Ali BodaghifardSajad Asadbegi Original Article 08 September 2015 Pages: 461 - 468
Functionalization of protected tyrosine via Sonogashira reaction: synthesis of 3-(1,2,3-triazolyl)-tyrosine Stanley N. S. VasconcelosAnwar ShamimHélio A. Stefani Original Article 26 October 2015 Pages: 469 - 481
One-pot tandem Ugi-4CR/\(\hbox {S}_{N}\)Ar approach to highly functionalized quino[2,3-b][1,5]benzoxazepines Mehdi GhandiNahid ZarezadehAlireza Abbasi Original Article 24 December 2015 Pages: 483 - 495
Facile synthesis and biological assays of novel 2,4-disubstituted hydrazinyl-thiazoles analogs Fateme Ghanbari PirbastiNosrat O. Mahmoodi Original Article 11 January 2016 Pages: 497 - 506
Simple and efficient synthesis of \(5'\)-aryl-\(5'\)-deoxyguanosine analogs by azide-alkyne click reaction and their antileishmanial activities Pierre DaligauxSébastien PomelChristian Cavé Original Article 11 January 2016 Pages: 507 - 519
Cathepsin D inhibitors as potential therapeutics for breast cancer treatment: Molecular docking and bioevaluation against triple-negative and triple-positive breast cancers Hasitha Shilpa AnantarajuMadhu Babu BattuPerumal Yogeeswari Original Article 13 November 2015 Pages: 521 - 535
High-throughput screening against \(\sim \)6.1 million structurally diverse, lead-like compounds to discover novel ROCK inhibitors for cerebral injury recovery Haoling GongZhicheng YuanLiping Zhan Original Article 23 December 2015 Pages: 537 - 549
Synthesis of tricyclic quinazolinones via intramolecular cyclization of 3-(2-aminoalkyl)-2-(phenylamino)quinazolin-4(3H)-ones Xuhong YangMinghu WuYalan Xing Short Communication 15 October 2015 Pages: 551 - 556
A green synthesis in water of novel (1,5,3-dithiazepan-3-yl)alkanoic acids by the multicomponent reaction of amino acids, \(\hbox {CH}_{2}\)O, and 1,2-ethanedithiol Guzel R. KhabibullinaEkaterina S. FedotovaAskhat G. Ibragimov Short Communication 29 January 2016 Pages: 557 - 565
Highly efficient synthesis of quinoxaline derivatives from 1,2-benzenediamine and \(\alpha \)-aminoxylated 1,3-dicarbonyl compounds Jianwei YanYanhong XuGuisheng Zhang Short Communication 21 January 2016 Pages: 567 - 573
Facile microwave-assisted synthesis of benzimidazole scaffolds via Ugi-type three-component condensation (3CC) reactions Gui-Ting SongZhi-Gang XuZhong-Zhu Chen Short Communication 18 November 2015 Pages: 575 - 580