1. Identification of furo[3′, 2′:3,4]naphtho[1,2-d]imidazole derivatives as orally active and selective inhibitors of microsomal prostaglandin E₂ synthase-1 (mPGES-1)

   • Chih-Hua Tseng
   • Cherng-Chyi Tzeng
   • Yeh-Long Chen

   Full-Length Paper 09 December 2011 Pages: 215 - 229

2. Combining click-multicomponent reaction: one-pot synthesis of triazolyl methoxy-phenyl indazolo[2,1-b]phthalazine-trione derivatives

   • Peyman Salehi
   • David I. MaGee
   • Jordan Donahue

   Full-Length Paper 11 December 2011 Pages: 231 - 240

3. Ionic liquid-supported synthesis of dihydroquinazolines and tetrahydroquinazolines under microwave irradiation

   • Hai-Yuan Hsu
   • Chih-Chun Tseng
   • Chung-Ming Sun

   Full-Length Paper 17 December 2011 Pages: 241 - 249

4. Synthesis, structure, and biological activity of novel (oxdi/tri)azoles derivatives containing 1,2,3-thiadiazole or methyl moiety

   • Xing-Hai Liu
   • Li Pan
   • Zheng-Ming Li

   Full-Length Paper 17 January 2012 Pages: 251 - 260

5. Generation of diverse 1-imidazolylisoquinolines via silver triflate-catalyzed reaction of 2-alkynylbenzaldoxime with imidazole

   • Qian Xiao
   • Shengqing Ye
   • Jie Wu

   Full-Length Paper 25 January 2012 Pages: 261 - 268

6. New approach for the synthesis of novel acenaphtho[1,2-b]furan-8-amines

   • Reza Sandaroos
   • Saman Damavandi
   • Maede Hasanpour

   Full-Length Paper 25 January 2012 Pages: 269 - 277

7. Intramolecular 1,3-dipolar cycloaddition reactions in the synthesis of complex annelated quinolines, α-carbolines and coumarins

   • Swarup Majumder
   • Pallabi Borah
   • Pulak J. Bhuyan

   Full-Length Paper 29 February 2012 Pages: 279 - 289

8. Synthesis of 5-alkylated barbituric acids and 3-alkylated indoles via microwave-assisted three-component reactions in solvent-free conditions using Hantzsch 1,4-dihydropyridines as reducing agents

   • Biswajita Baruah
   • P. Seetham Naidu
   • Pulak J. Bhuyan

   Full-Length Paper 02 February 2012 Pages: 291 - 298

9. Organocatalytic three-component cascade reaction for the synthesis of spiro[indeno[1,2-b]furan]-triones

   • Somayeh Ahadi
   • Maryam Abaszadeh
   • Ayoob Bazgir

   Full-Length Paper 15 March 2012 Pages: 299 - 306

10. Synthesis and in vitro inhibition properties of oligonucleotide conjugates carrying amphipathic proline-rich peptide derivatives of the sweet arrow peptide (SAP)

    • Santiago Grijalvo
    • Ramon Eritja

    Full-Length Paper 06 March 2012 Pages: 307 - 317

11. Task-specific nitrite and azide ionic liquids for the efficient one-pot synthesis of 1,2,3-triazoles from the aniline derivatives

    • Hassan Valizadeh
    • Mohammad Amiri
    • Elham Khalili

    Full-Length Paper 31 March 2012 Pages: 319 - 323

12. Diastereoselective multicomponent synthesis and anti-HSV-1 evaluation of dihydrofuran-fused derivatives

    • Angela Scala
    • Massimiliano Cordaro
    • Giovanni Grassi

    Full-Length Paper 22 April 2012 Pages: 325 - 333

13. Accessing a small library of pluripotent 1,4,5-trisubstituted 1H-1,2,3-triazoles via diversity-oriented synthesis

    • Arya Ajay
    • Munna Prasad Gupt
    • Rama P. Tripathi

    Full-Length Paper 22 April 2012 Pages: 335 - 350

14. A novel one-pot pseudo-five-component condensation reaction towards bifunctional diazepine-tetrazole containing compounds: synthesis of 1H-tetrazolyl-1H-1,4-diazepine-2,3-dicarbonitriles and 1H-tetrazolyl-benzo[b][1,4]diazepines

    • Hamid Mofakham
    • Ahmad Shaabani
    • Seik Weng Ng

    Full-Length Paper 17 May 2012 Pages: 351 - 356

15. Naturally occurring himachalenes to benzocycloheptene amino vinyl bromide derivatives: as antidepressant molecules

    • Abha Chaudhary
    • Pralay Das
    • Rajesh K. Goel

    Full-Length Paper 15 May 2012 Pages: 357 - 366

    

16. Scaffold hopping for identification of novel D₂ antagonist based on 3D pharmacophore modelling of illoperidone analogs

    • Radha Charan Dash
    • Sharad H. Bhosale
    • Kakasaheb R. Mahadik

    Full-Length Paper 08 December 2011 Pages: 367 - 375

17. 3D-QSAR and molecular docking analysis of biphenyl amide derivatives as p38α mitogen-activated protein kinase inhibitors

    • Pravin Sundarao Ambure
    • Rahul Prakashchand Gangwal
    • Abhay T. Sangamwar

    OriginalPaper 07 January 2012 Pages: 377 - 388

18. QSAR classification of metabolic activation of chemicals into covalently reactive species

    • Chin Yee Liew
    • Chuen Pan
    • Chun Wei Yap

    Full-Length Paper 28 February 2012 Pages: 389 - 400

19. Binding site characterization of G protein-coupled receptor by alanine-scanning mutagenesis using molecular dynamics and binding free energy approach: application to C-C chemokine receptor-2 (CCR2)

    • Swapnil Chavan
    • Shirishkumar Pawar
    • M. Elizabeth Sobhia

    Full-Length Paper 22 April 2012 Pages: 401 - 413

20. Synthesis of benzopyrano[4,3-b](N-arylsulfonyl)indoles and benzopyrano[3,4-b](N-arylsulfonyl)indoles via intramolecular palladium-catalyzed aryl–aryl coupling reaction

    • Ling-ling Fan
    • Zhi-ping Che
    • Hui Xu

    Short Communication 22 April 2012 Pages: 415 - 421