1. Conventional and microwave-assisted synthesis of new indole-tethered benzimidazole-based 1,2,3-triazoles and evaluation of their antimycobacterial, antioxidant and antimicrobial activities

   • Dongamanti Ashok
   • Srinivas Gundu
   • Mohan Gandhi Devulapally

   Original Article 18 April 2018 Pages: 769 - 778

   

2. Systematic search for benzimidazole compounds and derivatives with antileishmanial effects

   • Juan Carlos Sánchez-Salgado
   • Pablo Bilbao-Ramos
   • Yareli Rojas-Aguirre

   Original Article 10 May 2018 Pages: 779 - 790

   

3. Synthesis and three-dimensional quantitative structure-activity relationship study of quinazoline derivatives containing a 1,3,4-oxadiazole moiety as efficient inhibitors against Xanthomonas axonopodis pv. citri

   • Xiaobin Wang
   • Jinghua Yan
   • Wei Xue

   Original Article 28 May 2018 Pages: 791 - 802

   

4. Synthesis and biological evaluation of novel flavone/triazole/benzimidazole hybrids and flavone/isoxazole-annulated heterocycles as antiproliferative and antimycobacterial agents

   • Yerrabelly Jayaprakash Rao
   • Thummala Sowjanya
   • Sudha Sravanti Kotapalli

   Original Article 04 June 2018 Pages: 803 - 814

   

5. New 7-piperazinylquinolones containing (benzo[d]imidazol-2-yl)methyl moiety as potent antibacterial agents

   • Hojat-Allah Arab
   • Mohammad Ali Faramarzi
   • Saeed Emami

   Original Article 07 June 2018 Pages: 815 - 825

   

6. Synthesis, docking and anticancer activity of azo-linked hybrids of 1,3,4-thia-/oxadiazoles with cyclic imides

   • Priyanka Bhatt
   • Manoj Kumar
   • Anjali Jha

   Original Article 08 June 2018 Pages: 827 - 840

   

7. Synthesis, in vitro \(\alpha \)-glucosidase inhibitory activity, and in silico study of (E)-thiosemicarbazones and (E)-2-(2-(arylmethylene)hydrazinyl)-4-arylthiazole derivatives

   • Muhammad Ali
   • Khalid Mohammed Khan
   • Shahnaz Perveen

   Original Article 29 May 2018 Pages: 841 - 861

   

8. Highly efficient synthesis of alkyl and aryl primary thiocarbamates and dithiocarbamates under metal- and solvent-free conditions

   • Ali Reza Sardarian
   • Iman Dindarloo Inaloo
   • Ali Reza Modarresi-Alam

   Original Article 12 June 2018 Pages: 863 - 878

   

9. One-pot synthesis of biologically active 1,2,3-trisubstituted pyrrolo[2,3-b]quinoxalines through a palladium-catalyzed reaction with internal alkyne moieties

   • Ali Keivanloo
   • Tayebeh Besharati-Seidani
   • Tsutomu Yokomatsu

   Original Article 16 June 2018 Pages: 879 - 891

   

10. Structure–activity relationship investigation of coumarin–chalcone hybrids with diverse side-chains as acetylcholinesterase and butyrylcholinesterase inhibitors

    • Lu Kang
    • Xiao-Hui Gao
    • Jian-Ye Yan

    Original Article 22 June 2018 Pages: 893 - 906

    

11. Regioselective four-component synthesis of new tetrazolo[1,5-a]quinoline-based 2-amino-1,4-dihydropyridine and pyridin-2(1H)-one derivatives using nano-ZnO catalysis

    • Tooran Aghaalizadeh
    • Farough Nasiri

    Original Article 27 June 2018 Pages: 907 - 917

    

12. 4-Amino-2,3-dihydro-1λ⁶-isothiazole-1,1-dioxides and their chemical properties evaluation

    • Maksim S. Dyachenko
    • Alexey V. Dobrydnev
    • Yulian M. Volovenko

    Original Article 28 June 2018 Pages: 919 - 927

    

13. Insights into the interaction and binding mode of a set of antifungal azoles as inhibitors of potential fungal enzyme-based targets

    • Camilo Guerrero-Perilla
    • Freddy A. Bernal
    • Ericsson Coy-Barrera

    Original Article 29 June 2018 Pages: 929 - 942

    

14. One-pot synthesis, biological evaluation and molecular docking studies of fused thiazolo[2,3-b]pyrimidinone-pyrazolylcoumarin hybrids

    • Ramesh Gondru
    • Saikiran Reddy Peddi
    • Rajitha Bavantula

    Original Article 02 July 2018 Pages: 943 - 956

    

15. Synthesis of new chiral 1,3,4-thiadiazole-based di- and tri-arylsulfonamide residues and evaluation of in vitro anti-HIV activity and cytotoxicity

    • Maria Shafique
    • Shahid Hameed
    • Najim Aboud Al-Masoudi

    Original Article 02 July 2018 Pages: 957 - 968

    

16. An efficient and facile synthesis of new tetracyclic fused pyrazolo[4,3-c][1,2,4]triazino[4,5-a]quinolin-4(5H)-ones

    • Mohsen A.-M. Gomaa
    • Huda A. Ali

    Original Article 03 July 2018 Pages: 969 - 977

    

17. ADME properties evaluation in drug discovery: in silico prediction of blood–brain partitioning

    • Lu Zhu
    • Junnan Zhao
    • Haichun Liu

    Original Article 06 August 2018 Pages: 979 - 990

    

18. Dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-4-ones as a new class of CK2 inhibitors

    • Mykola V. Protopopov
    • Olga V. Ostrynska
    • Sergiy M. Yarmoluk

    Short Communication 29 May 2018 Pages: 991 - 998

    

19. Synthesis of some new triamide derivatives via Ugi five-component reaction in aqueous solution

    • Ali Asghar Mohammadi
    • Salman Taheri
    • Reza Ahdenov

    Short Communication 27 June 2018 Pages: 999 - 1006