1. Privileged heterocyclic scaffolds in chemical biology and drug discovery: synthesis and bioactivity

   News 27 April 2017 Pages: 239 - 239

   

2. N-(Hetero)aryl-2-imidazolines: an emerging privileged motif for contemporary drug design

   • Mikhail Krasavin

   REVIEWS 26 April 2017 Pages: 240 - 255

   

3. Preparation and biological properties of 2-thio-containing pyrimidines and their condensed analogs

   • Oleksii Yu. Voskoboynik
   • Oleksandra S. Kolomoets
   • Sergiy I. Kovalenko

   OriginalPaper 27 April 2017 Pages: 256 - 272

   

4. Heterocycles as classical and nonclassical ring B isosters in combretastatin A-4

   • Nikolay A. Zefirov
   • Olga N. Zefirova

   OriginalPaper 24 April 2017 Pages: 273 - 280

   

5. 1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents

   • Giulia Venditti
   • Giovanna Poce
   • Mariangela Biava

   OriginalPaper 27 April 2017 Pages: 281 - 291

   

6. 2-(Azolyl)anilines: methods of synthesis, cyclocondensations, and biological properties

   • Oleksii M. Antypenko
   • Sergiy V. Kholodnyak
   • Sergiy I. Kovalenko

   OriginalPaper 25 April 2017 Pages: 292 - 309

   

7. 3,4-Dihydroquinoxalin-2-ones: recent advances in synthesis and bioactivities (microreview)

   • Tone Kristoffersen
   • Jørn H. Hansen

   HETEROCYCLES IN FOCUS 26 April 2017 Pages: 310 - 312

   

8. Synthesis of indolizinium salts (microreview)

   • Anna Ivanova
   • Pavel Arsenyan

   HETEROCYCLES IN FOCUS 24 April 2017 Pages: 313 - 315

   

9. Exploring the influence of the substituent at position 4 in a series of 3,4-dihydropyrimidin-2(1H)-one A_2B adenosine receptor antagonists

   • Abel Crespo
   • Abdelaziz El Maatougui
   • Eddy Sotelo

   OriginalPaper 26 April 2017 Pages: 316 - 321

   

10. Functionalization of four-membered cyclic sulfoximines by a convenient lithiation/trapping sequence

    • Arianna Tota
    • Flavio Fanelli
    • Leonardo Degennaro

    OriginalPaper 27 April 2017 Pages: 322 - 328

    

11. 2-Arylazetidines as ligands for nicotinic acetylcholine receptors

    • Leonardo Degennaro
    • Marina Zenzola
    • Giovanni Lentini

    OriginalPaper 26 April 2017 Pages: 329 - 334

    

12. Synthesis and structure of dihydroberberine nitroaryl derivatives – potential ligands for G-quadruplexes

    • Oleg N. Burov
    • Sergey V. Kurbatov
    • Igor E. Mikhailov

    OriginalPaper 26 April 2017 Pages: 335 - 340

    

13. Investigation on the synthesis of new 3-[4-(arylalkoxy)phenylethyl]-2-thioxo-1,3-thiazolidin-4-ones and their biological evaluation against cancer cells

    • Camille Déliko Dago
    • Christelle N’ta Ambeu
    • Jean-Pierre Bazureau

    OriginalPaper 27 April 2017 Pages: 341 - 349

    

14. Synthesis of phenylpyridine derivatives and their biological evaluation toward dipeptidyl peptidase-4

    • Yan Zhu
    • Xiangguo Meng
    • Weicheng Zhou

    OriginalPaper 26 April 2017 Pages: 350 - 356

    

15. Physicochemical properties and antimicrobial activity of new spirocyclic thieno[2,3-d]pyrimidin-4(3H)-one derivatives

    • Modesto de Candia
    • Claudia Altamura
    • Cosimo D. Altomare

    OriginalPaper 27 April 2017 Pages: 357 - 363

    

16. Synthesis of new heterocyclic dehydroabietylamine derivatives and their biological activity

    • Kseniya S. Kovaleva
    • Olga I. Yarovaya
    • Nariman F. Salakhutdinov

    OriginalPaper 27 April 2017 Pages: 364 - 370

    

17. Synthesis and biological activity of heterocyclic borneol derivatives

    • Anastasiya S. Sokolova
    • Olga I. Yarovaya
    • Nariman F. Salakhutdinov

    OriginalPaper 24 April 2017 Pages: 371 - 377

    

18. (5S,7R)-5-Aryl-7-methyl-4,5,6,7-tetrahydro-[1, 2, 4]triazolo[1,5-a]pyrimidin-7-ols as products of three-component condensation

    • Sergey A. Komykhov
    • Andrey A. Bondarenko
    • Sergey M. Desenko

    SHORT COMMUNICATION 22 April 2017 Pages: 378 - 380