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Fluoro-containing Heterocycles: XIII. Fluoro-containing Derivatives of Thiazolo[3,2-a]-, Benzothiazolo[3,2-a]-, and Benzimidazo[3,2-a]quinazolinones

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Abstract

Reactions of 2-aminothiazole, derivatives of 2-aminobenzothiazole and 2-aminobenzoimidazole with polyfluorobenzoyl chlorides gave rise to acylation products that at heating in the diphenyl ether formed fluoro-containing derivatives of thiazolo[3,2-a]-, benzothiazolo[3,2-a]-, and benzimidazo[3,2-a]quinazolinone.

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Authors and Affiliations

  1. Ural State Technical University, Yekaterinburg, 620002, Russia

    E. V. Nosova, G. N. Lipunova, A. A. Laeva & V. N. Charushin

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  1. E. V. Nosova
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  2. G. N. Lipunova
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  3. A. A. Laeva
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  4. V. N. Charushin
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__________

Translated from Zhurnal Organicheskoi Khimii, Vol. 41, No. 11, 2005, pp. 1705–1711.

Original Russian Text Copyright © 2005 by Nosova, Lipunova, Laeva, Charushin.

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Nosova, E.V., Lipunova, G.N., Laeva, A.A. et al. Fluoro-containing Heterocycles: XIII. Fluoro-containing Derivatives of Thiazolo[3,2-a]-, Benzothiazolo[3,2-a]-, and Benzimidazo[3,2-a]quinazolinones. Russ J Org Chem 41, 1671–1677 (2005). https://doi.org/10.1007/s11178-006-0017-9

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  • DOI: https://doi.org/10.1007/s11178-006-0017-9

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