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Synthesis and anxiolytic activity of 2-aminoadamantane derivatives containing monoterpene fragments

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Two new amines were synthesized from 2-aminoadamantane and the available monoterpenoid aldehydes citral and (–)-myrtenal. It was established that the synthesized amines possessed anxiolytic activity.

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Correspondence to E. V. Suslov.

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Translated from Khimiko-Farmatsevticheskii Zhurnal, Vol. 46, No. 5, pp.3–5, May, 2012.

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Kapitsa, I.G., Suslov, E.V., Teplov, G.V. et al. Synthesis and anxiolytic activity of 2-aminoadamantane derivatives containing monoterpene fragments. Pharm Chem J 46, 263–265 (2012). https://doi.org/10.1007/s11094-012-0775-3

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  • DOI: https://doi.org/10.1007/s11094-012-0775-3

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