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Synthesis, antiviral and antimicrobial screening of some new 2-oxoindoline derivatives

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Chemistry of Heterocyclic Compounds Aims and scope

New 3-(2-(5-(aryldiazenyl)-4-methylthiazol-2-yl)hydrazono)indolin-2-ones were prepared by the reaction of isatin β-thiosemicarbazone with different hydrazonoyl chlorides. Imide derivatives were prepared by the reaction of isatin hydrazone with various anhydrides, and a series of new sulfonimides was also synthesized. All new compounds were tested for their biological activities.

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Authors and Affiliations

  1. Applied Organic Chemistry Department, National Research Center, Dokki, Giza, Egypt

    Madiha Farghaly & Bakr F. Abdel-Wahab

  2. Natural and Microbial Products Chemistry Department, National Research Center, Dokki, Giza, Egypt

    Essam M. Ahmed

Authors
  1. Madiha Farghaly
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  2. Bakr F. Abdel-Wahab
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  3. Essam M. Ahmed
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Corresponding author

Correspondence to Bakr F. Abdel-Wahab.

Additional information

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 5, pp. 689-694, May, 2009.

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Farghaly, M., Abdel-Wahab, B.F. & Ahmed, E.M. Synthesis, antiviral and antimicrobial screening of some new 2-oxoindoline derivatives. Chem Heterocycl Comp 45, 539–544 (2009). https://doi.org/10.1007/s10593-009-0301-z

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  • DOI: https://doi.org/10.1007/s10593-009-0301-z

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