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Synthesis andin vitro cytotoxicity of 1-azaanthraquinone-3-carboxamides

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Abstract

Five 1-azaanthraquinone-3-carboxamides were synthesized and evaluated in vitro cytotoxicity against four human cancer cell lines. The most active compound,7b, exhibited cytotoxic activity comparable to doxorubicin.

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Correspondence to Heesoon Lee.

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Lee, H., Lee, Cw. & Yang, SI. Synthesis andin vitro cytotoxicity of 1-azaanthraquinone-3-carboxamides. Arch Pharm Res 22, 380–383 (1999). https://doi.org/10.1007/BF02979061

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