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Synthetic combinatorial libraries: Views on techniques and their application

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Perspectives in Drug Discovery and Design

Summary

This paper reviews synthetic combinatorial libraries. Particular emphasis is placed on one-bead-one-compound libraries, although issues relating to all synthetic techniques are touched upon. The discussion is focused on questions relating to synthetic diversity, drug discovery assays and structure determination techniques.

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  1. Selectide Corporation, 1580 E. Hanley Boulevard, 85737, Tucson, AZ, USA

    Dave Madden, Viktor Krchňák & Michael Lebl

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  2. Viktor Krchňák
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Madden, D., Krchňák, V. & Lebl, M. Synthetic combinatorial libraries: Views on techniques and their application. Perspectives in Drug Discovery and Design 2, 269–285 (1995). https://doi.org/10.1007/BF02172067

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