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Lisuride and [C-11]-Raclopride Interaction at the D2 Receptor Site

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PET for Drug Development and Evaluation

Part of the book series: Developments in Nuclear Medicine ((DNUM,volume 26))

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Abstract

Dopaminergic drugs exert their action through activation of dopamine D1 and D2 receptors [1]. Changes of dopamine receptor density or affinity following antiparkinsonian drug therapy is suggested to underlie the development of long-term treatment complications in patients with PD [2]. However, evidence for this has not been provided.

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References

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© 1995 Springer Science+Business Media Dordrecht

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Leenders, K.L., Antonini, A. (1995). Lisuride and [C-11]-Raclopride Interaction at the D2 Receptor Site. In: Comar, D. (eds) PET for Drug Development and Evaluation. Developments in Nuclear Medicine, vol 26. Springer, Dordrecht. https://doi.org/10.1007/978-94-011-0429-6_19

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  • DOI: https://doi.org/10.1007/978-94-011-0429-6_19

  • Publisher Name: Springer, Dordrecht

  • Print ISBN: 978-94-010-4191-1

  • Online ISBN: 978-94-011-0429-6

  • eBook Packages: Springer Book Archive

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