Preparation, Reactivity, and Synthetic Utility of Simple Benzotriazole Derivatives

  • Romaric Gérardy
  • Jean-Christophe M. MonbaliuEmail author
Part of the Topics in Heterocyclic Chemistry book series (TOPICS, volume 43)


The benzotriazole fragment is known to behave as (1) an excellent leaving group, (2) an electron-donating or an electron-withdrawing group, (3) an anion precursor, and (4) a radical precursor. It confers unique physicochemical properties to its immediate vicinity on various molecular scaffolds. This review covers the preparation and synthetic utility of versatile benzotriazole derivatives. The selected compounds are conveniently prepared from 1H-benzotriazole and are characterized by a huge synthetic potential. Their specific reactivity is discussed and illustrated with various examples ranging from methodology in organic chemistry to the total synthesis of complex structures.


Benzotriazole derivatives Benzotriazole methodology Molecular diversity Versatile synthons 


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Copyright information

© Springer International Publishing Switzerland 2015

Authors and Affiliations

  • Romaric Gérardy
    • 1
  • Jean-Christophe M. Monbaliu
    • 1
    Email author
  1. 1.Center for Integrated Technology and Organic Synthesis, Department of ChemistryUniversity of LiègeLiègeBelgium

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