Abstract
Number of novel derivatives of dihydrotriazolo-and-tetrazolopyrimidines containing carboxamide group in position 6 were obtained by multicomponent Biginelli-type reaction. The structures of all synthesized compounds were proved by NMR and MS spectral methods. The method of three-component Biginelli-type reaction is well suited for the synthesis of new promising dihydroazolopyrimidines providing a scaffold for screening of biological activity.
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Gladkov, E., Sirko, S., Khanetskii, B. et al. Multicomponent facile synthesis of novel dihydroazolopyrimidinyl carbamides. Chem. Pap. 61, 146–149 (2007). https://doi.org/10.2478/s11696-007-0012-9
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DOI: https://doi.org/10.2478/s11696-007-0012-9