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An Easy, Efficient and Improved Synthesis of Sertaconazole Nitrate

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Abstract

An easy, efficient and improved synthetic route has been developed for the synthesis of Sertaconazole (1-{2-[(7-chlorobenzo[b]thiophen-3-yl)methoxy]-2-(2,4-dichlorophenyl)ethyl}-1H-imidazole) employing multiple chemical transformation.

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Acknowledgments

The authors wish to thank Dr. V.V.S.V Prasad and Dr. Dipankar Karmakar for their valuable support.

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Authors and Affiliations

  1. Department of Research and Development, Seutic Labs Private Limited, Jeedimetla, Hyderabad, Telangana, 500055, India

    S. Venkateswarlu Rayudu

  2. Centre for Chemical Sciences, Institute of Science and Technology, Jawaharlal Nehru Technological University, Kukatpally, Hyderabad, Telangana, 500072, India

    S. Venkateswarlu Rayudu & P. Kumar

Authors
  1. S. Venkateswarlu Rayudu
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  2. P. Kumar
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Corresponding author

Correspondence to S. Venkateswarlu Rayudu.

Additional information

Russian Text © The Author(s), 2019, published in Zhurnal Organicheskoi Khimii, 2019, Vol. 55, No. 8, pp. 1310.

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Venkateswarlu Rayudu, S., Kumar, P. An Easy, Efficient and Improved Synthesis of Sertaconazole Nitrate. Russ J Org Chem 55, 1212–1216 (2019). https://doi.org/10.1134/S1070428019080219

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  • DOI: https://doi.org/10.1134/S1070428019080219

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