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Synthesis of hetarylquinolines proceeding from 2-[(2-methylquinolin-4-yl)sulfanyl]acetohydrazide substituted in the benzene ring

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Abstract

At intramolecular cyclization of phenylhydrazinocarbothioamide in alkaline and acidic media quinolyl-substituted triazoles and thiadiazoles are obtained. Quinolyl-substituted thiazolidines and thiazolidinones were obtained at interaction of phenylhydrazinocarbothioamides with bromoacetophenone and ethyl bromoacetate.

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Authors and Affiliations

  1. Yerevan State University, ul. Aleka Manukyana 1, Yerevan, 375025, Armenia

    I. L. Aleksanyan & L. P. Hambardzumyan

Authors
  1. I. L. Aleksanyan
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  2. L. P. Hambardzumyan
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Correspondence to I. L. Aleksanyan.

Additional information

Original Russian Text © I.L. Aleksanyan, L.P. Hambardzumyan, 2017, published in Zhurnal Organicheskoi Khimii, 2017, Vol. 53, No. 2, pp. 233–236.

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Aleksanyan, I.L., Hambardzumyan, L.P. Synthesis of hetarylquinolines proceeding from 2-[(2-methylquinolin-4-yl)sulfanyl]acetohydrazide substituted in the benzene ring. Russ J Org Chem 53, 226–230 (2017). https://doi.org/10.1134/S1070428017020142

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  • DOI: https://doi.org/10.1134/S1070428017020142

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