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Synthesis of a triterpene-spermidine conjugate

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Abstract

Three synthetic approaches to triterpene-spermidine conjugate coupled at the C3 atom have been tested. The best yield was obtained by reductive amination of betulonic acid methyl ester with spermidine.

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Authors and Affiliations

  1. Institute of Organic Chemistry, Ufa Research Center, Russian Academy of Sciences, pr. Oktyabrya 71, Ufa, 450054, Bashkortostan, Russia

    O. B. Kazakova, G. V. Giniyatullina, N. I. Medvedeva & G. A. Tolstikov

Authors
  1. O. B. Kazakova
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  2. G. V. Giniyatullina
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  3. N. I. Medvedeva
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  4. G. A. Tolstikov
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Corresponding author

Correspondence to O. B. Kazakova.

Additional information

Original Russian Text © O.B. Kazakova, G.V. Giniyatullina, N.I. Medvedeva, G.A. Tolstikov, 2012, published in Zhurnal Organicheskoi Khimii, 2012, Vol. 48, No. 10, pp. 1370–1373.

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Kazakova, O.B., Giniyatullina, G.V., Medvedeva, N.I. et al. Synthesis of a triterpene-spermidine conjugate. Russ J Org Chem 48, 1366–1369 (2012). https://doi.org/10.1134/S1070428012100181

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  • DOI: https://doi.org/10.1134/S1070428012100181

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