Abstract
A new synthetic approach was developed to the preparation of functional derivatives of 3-(1,3,4-oxadiazol-2-yl)-1H-indoles starting with a synthetically available 3-[5-(chloromethyl)-1,3,4-oxadiazol-2-yl]-1H-indole. The versatility of the developed strategy was demonstrated in the synthesis of this kind compounds with a wide range of substituents.
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Original Russian Text © S.B. Alyab’ev, D.V. Kravchenko, A.V. Ivashchenko, 2009, published in Zhurnal Organicheskoi Khimii, 2009, Vol. 45, No. 5, pp. 734–739.
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Alyab’ev, S.B., Kravchenko, D.V. & Ivashchenko, A.V. Functionalization of oxadiazolylindole systems. Russ J Org Chem 45, 719–724 (2009). https://doi.org/10.1134/S1070428009050121
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DOI: https://doi.org/10.1134/S1070428009050121