Skip to main content
Log in

Functionalization of oxadiazolylindole systems

  • Published:
Russian Journal of Organic Chemistry Aims and scope Submit manuscript

Abstract

A new synthetic approach was developed to the preparation of functional derivatives of 3-(1,3,4-oxadiazol-2-yl)-1H-indoles starting with a synthetically available 3-[5-(chloromethyl)-1,3,4-oxadiazol-2-yl]-1H-indole. The versatility of the developed strategy was demonstrated in the synthesis of this kind compounds with a wide range of substituents.

This is a preview of subscription content, log in via an institution to check access.

Access this article

Price excludes VAT (USA)
Tax calculation will be finalised during checkout.

Instant access to the full article PDF.

Similar content being viewed by others

References

  1. Biradar, J.S. and Manjunath, S.Y., Indian J. Chem. B, 2004, vol. 43, p. 141.

    Google Scholar 

  2. Swain, C.J., Baker, R., Kneen, C., Moseley, J., Saunders, J., Seward, E.M., Stevenson, G., Beer, M., Stanton, J., Watling, K., J. Med. Chem., 1991, vol. 34, p. 140.

    Article  CAS  Google Scholar 

  3. Danawade, D.S., Raghu, A.V., and Gadaginamath, G.S., Indian J. Chem. B, 2006, vol. 45, p. 689.

    Google Scholar 

  4. Ushakova, R.L., Mikaya, A.I., Zaikin, V.G., Kelarev, V.I., and Shvekhgeimer, G.A., Khim. Geterotsikl. Soedin., 1986, vol. 22, p. 539.

    Google Scholar 

  5. Kelarev, V.I. and Shvekhgeimer, G.A., Khim. Geterotsikl. Soedin., 1982, p. 343.

  6. Kelarev, V.I. and Shvekhgeimer, G.A., Izv. Vuzov, Ser. Khim. i, Khim. Tekhnol., 1982, vol. 25, p. 1458.

    CAS  Google Scholar 

  7. Kelarev, V.I, Gasanov, S.Sh., Karakhanov, R.A., Polivin, Yu.N., Kuatbekova, K.P., and Panina, M.E., Zh. Org. Khim., 1992, vol. 28, p. 2561.

    CAS  Google Scholar 

  8. Farghaly, Abdel-Rahman, A.H., J. Chin. Chem. Soc., 2004, vol. 51, p. 147.

    Google Scholar 

  9. Ottoni, O., Cruz, R., and Alves, R. Tetrahedron, 1998, vol. 54, p. 13915.

    Article  CAS  Google Scholar 

Download references

Author information

Authors and Affiliations

Authors

Corresponding author

Correspondence to S. B. Alyab’ev.

Additional information

Original Russian Text © S.B. Alyab’ev, D.V. Kravchenko, A.V. Ivashchenko, 2009, published in Zhurnal Organicheskoi Khimii, 2009, Vol. 45, No. 5, pp. 734–739.

Rights and permissions

Reprints and permissions

About this article

Cite this article

Alyab’ev, S.B., Kravchenko, D.V. & Ivashchenko, A.V. Functionalization of oxadiazolylindole systems. Russ J Org Chem 45, 719–724 (2009). https://doi.org/10.1134/S1070428009050121

Download citation

  • Received:

  • Published:

  • Issue Date:

  • DOI: https://doi.org/10.1134/S1070428009050121

Keywords

Navigation