Abstract
Electrophilic intramolecular heterocyclization of 3-(2-chloroprop-2-en-1-yl)-2-methylquinolin-4-ol by the action of bromine gave 2-bromomethyl-2-chloro-4-methyl-2,3-dihydrofuro[3,2-c]quinoline hydrobromide which was converted into 2-hydroxymethyl-, 2-alkoxymethyl-, and 2-dialkylaminomethyl-4-methylfuro[3,2-c]quinolines by treatment with the corresponding nucleophiles.
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Original Russian Text © A.A. Avetisyan, I.L. Aleksanyan, K.S. Sargsyan, 2007, published in Zhurnal Organicheskoi Khimii, 2007, Vol. 43, No. 3, pp. 427–429.
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Avetisyan, A.A., Aleksanyan, I.L. & Sargsyan, K.S. Synthesis of 2-bromomethyl-4-methyl-2,3-dihydrofuro[3,2-c]-quinoline and some its transformations. Russ J Org Chem 43, 426–428 (2007). https://doi.org/10.1134/S1070428007030177
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DOI: https://doi.org/10.1134/S1070428007030177