Russian Journal of General Chemistry

, Volume 88, Issue 4, pp 676–681 | Cite as

Synthesis and Antibacterial Activity of 9-Oxo-9,10-dihydroacridinecarboxylic Acids Esters Bearing a Triazole Fragment

  • T. N. Kudryavtseva
  • A. Yu. Lamanov
  • L. G. Klimova
  • G. V. Nazarov


An effective method for the synthesis of new acridine-9(10H)-one (acridone) derivatives containing 1,2,3-triazole fragment was developed. A number of new triazole-containing compounds were synthesized from propargyl acridone acetate and their antimicrobial activity was studied.


acridone triazole nitrofuran antibacterial activity 


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This work was financially supported by the Ministry of Education and Science of Russia (project no. 4.9516.2017/BCh).


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Copyright information

© Pleiades Publishing, Ltd. 2018

Authors and Affiliations

  • T. N. Kudryavtseva
    • 1
  • A. Yu. Lamanov
    • 1
  • L. G. Klimova
    • 2
  • G. V. Nazarov
    • 1
  1. 1.Kursk State UniversityKurskRussia
  2. 2.Kursk State Medical UniversityKurskRussia

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