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Russian Journal of General Chemistry

, Volume 88, Issue 2, pp 334–337 | Cite as

Synthesis of 4-Aryl-2-hydroxy-4-oxo-N-{4-[(1,3-thiazol-2-yl)- sulfamoyl]phenyl}but-2-eneamides

  • V. L. Gein
  • O. V. Bobrovskaya
  • A. A. Russkikh
  • N. N. Petukhova
Letters to the Editor
  • 33 Downloads

Abstract

The reaction of methyl aroylpyruvates with 2-(4-aminobenzenesulfamido)thiazole (norsulfazole) in glacial acetic acid in the presence of anhydrous sodium acetate furnished 4-aryl-2-hydroxy-4-oxo-N-{4-[(1,3-thiazol-2-yl)sulfamoyl]phenyl}but-2-eneamides.

Keywords

4-aryl-2-hydroxy-4-oxo-N-{4-[(1,3-thiazol-2-yl)sulfamoyl]phenyl}but-2-eneamides 2-(4-aminobenzenesulfamido) thiazole norsulfazole 

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Copyright information

© Pleiades Publishing, Ltd. 2018

Authors and Affiliations

  • V. L. Gein
    • 1
  • O. V. Bobrovskaya
    • 1
  • A. A. Russkikh
    • 1
  • N. N. Petukhova
    • 1
  1. 1.Perm State Pharmaceutical AcademyPermRussia

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