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Synthesis of 2-aryl-4-cyano-1,3-oxazole-5-sulfonyl chlorides and N-substituted sulfonamides

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Abstract

Oxidative chlorination of 2-aryl-5-benzylsulfanyl-1,3-oxazole-4-carbonitrile results in the previously unknown 4-cyano-1,3-oxazole-5-sulfonyl chlorides and N-substituted sulfonamides.

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Authors and Affiliations

  1. Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine, ul. Murmanskaya 1, Kiev-94, 02660, Ukraine

    A. N. Kornienko, S. G. Pil’o, V. M. Prokopenko & V. S. Brovarets

Authors
  1. A. N. Kornienko
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  2. S. G. Pil’o
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  3. V. M. Prokopenko
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  4. V. S. Brovarets
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Corresponding author

Correspondence to V. S. Brovarets.

Additional information

Original Russian Text © A.N. Kornienko, S.G. Pil’o, V.M. Prokopenko, V.S. Brovarets, 2012, published in Zhurnal Obshchei Khimii, 2012, Vol. 82, No. 11, pp. 1865–1869.

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Kornienko, A.N., Pil’o, S.G., Prokopenko, V.M. et al. Synthesis of 2-aryl-4-cyano-1,3-oxazole-5-sulfonyl chlorides and N-substituted sulfonamides. Russ J Gen Chem 82, 1855–1858 (2012). https://doi.org/10.1134/S1070363212110229

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  • DOI: https://doi.org/10.1134/S1070363212110229

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