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Russian Journal of Organic Chemistry

, Volume 54, Issue 8, pp 1241–1249 | Cite as

Synthesis and Chemical Transformations of 5-Alkyl(phenyl)-4,5,6,7-tetrahydro[1,2,4]triazolo[1,5-a]pyrimidin-7-oles

  • N. I. Zemlyanaya
  • T. M. Karnozhitskaya
  • V. I. Musatov
  • I. S. Konovalova
  • S. V. Shishkina
  • V. V. Lipson
Article
  • 3 Downloads

Abstract

5,5,7-Trimethyl-4,5,6,7-tetrahydro[1,2,4]triazolo[1,5-a]pyrimidin-7-ol was synthesized by cyclocondensation of 3-amino-1,2,4-triazole with 4-methylpent-3-en-2-one; its chemical transformations, and also the transformations of 5-phenyl-4,5,6,7-tetrahydro[1,2,4]triazolo[1,5-a]pyrimidin-7-ol were investigated in reactions with reagents of diverse electronic nature.

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Copyright information

© Pleiades Publishing, Ltd. 2018

Authors and Affiliations

  • N. I. Zemlyanaya
    • 1
    • 2
  • T. M. Karnozhitskaya
    • 1
  • V. I. Musatov
    • 2
  • I. S. Konovalova
    • 2
  • S. V. Shishkina
    • 2
    • 3
  • V. V. Lipson
    • 1
    • 2
    • 3
  1. 1.Danilevsky Institute of Problems of Endocrine PathologyNational Academy of Sciences of UkraineKharkivUkraine
  2. 2.Institute of Single CrystalsNational Academy of Sciences of UkraineKharkivUkraine
  3. 3.Karazin Kharkiv National UniversityKharkivUkraine

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