Abstract
Ugi reaction with 5-isocyanoindoles afforded a number of amino acids, β-lactams, and tetrazoles. The described approach can be applied to combinatorial synthesis of biologically active compounds of the indole series.
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Mironov, M.A., Tokareva, M.I., Ivantsova, M.N. et al. Ugi Reaction with Isocyanoindoles. Russian Journal of Organic Chemistry 40, 847–853 (2004). https://doi.org/10.1023/B:RUJO.0000044548.07660.3c
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DOI: https://doi.org/10.1023/B:RUJO.0000044548.07660.3c