Abstract
Radioiodination of tri-n-butylstannyl-3-quinuclidinyl benzilate (TQNB) and N-succinimidyl-3-(tri-n-butylstannyl) benzoate (STB) was studied. STB was radiolabeled efficiently using iodogen to prepare radioactive N-succinimidyl-3- iodobenzoate (S125IB). TQNB was radioiodinated using Chloramine-T to obtain radioactive iodo-3-quinuclidinyl benzilate (125IQNB). Both S125IB and 125IQNB showed good stability at room temperature in the dark.
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Wang, L.H., Wang, Y.X., Yin, D.Z. et al. Radioiodination of aromatic organostannates. Journal of Radioanalytical and Nuclear Chemistry 258, 685–688 (2003). https://doi.org/10.1023/B:JRNC.0000011771.46058.6a
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DOI: https://doi.org/10.1023/B:JRNC.0000011771.46058.6a