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Conversion of Epiandrosterone Into 17β-Amino-5α-androstane

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Abstract

A new method for synthesizing 17β-amino-5α-androstane was developed based on tigogenin. The configuration at C-17 was proved by PMR.

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Authors and Affiliations

  1. I. G. Kutateladze Institute of Pharmaceutical Chemistry, Academy of Sciences of Georgia, Tbilisi, 0159, ul. Saradzhishvili 36

    M. I. Merlani, M. G. Davitishvili, N. Sh. Nadaraia & M. I. Sikharulidze

  2. Institute of Physical Chemistry, National Scientific-Research Center DEMOKRITOS, Athens, Greece

    K. Papadopulos

Authors
  1. M. I. Merlani
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  2. M. G. Davitishvili
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  3. N. Sh. Nadaraia
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  4. M. I. Sikharulidze
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  5. K. Papadopulos
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Merlani, M.I., Davitishvili, M.G., Nadaraia, N.S. et al. Conversion of Epiandrosterone Into 17β-Amino-5α-androstane. Chemistry of Natural Compounds 40, 144–146 (2004). https://doi.org/10.1023/B:CONC.0000033931.36367.0d

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  • DOI: https://doi.org/10.1023/B:CONC.0000033931.36367.0d

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