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Nitriles in Organic Synthesis: Synthesis of Pyrido[2,1-b]benzothiazole Derivatives and Polyfunctionally-substituted Pyridines

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

A variety of pyrido[2,1-b]benzothiazole derivatives could be prepared by reaction of 2-cyanomethylbenzothiazole, formaldehyde, and various active methylene reagents. Also some polyfunctionally-substituted pyridines were prepared by reaction of 2-cyanomethylbenzothiazole, formaldehyde, and an α-functionally substituted acrylonitrile.

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Authors and Affiliations

  1. Photochemistry Department, National Research Center, Dokki, Cairo, Egypt

    M. E. A. Zaki

  2. Chemistry Department, Faculty of Science, Mansoura University, Mansoura, Egypt

    A. A. Fadda, K. Samir & F. A. Amer

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  1. M. E. A. Zaki
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  2. A. A. Fadda
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  3. K. Samir
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  4. F. A. Amer
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Zaki, M.E.A., Fadda, A.A., Samir, K. et al. Nitriles in Organic Synthesis: Synthesis of Pyrido[2,1-b]benzothiazole Derivatives and Polyfunctionally-substituted Pyridines. Chemistry of Heterocyclic Compounds 39, 1242–1248 (2003). https://doi.org/10.1023/B:COHC.0000008274.04008.c2

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  • DOI: https://doi.org/10.1023/B:COHC.0000008274.04008.c2

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