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A new approach to CF3-containing 3,4-dihydroquinazolin-2(1H)-ones

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Abstract

A new approach to CF3-containing 3,4-dihydroquinazolin-2(1H)-ones based on the condensation of 5-acetyl-6-methyl-1-phenyl-4-trifluoromethylpyrimidin-2(1H)-one with dimethylformamide dimethyl acetal has been suggested.

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Authors and Affiliations

  1. N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991, Moscow, Russian Federation

    L. S. Vasil’ev, S. V. Baranin, A. S. Dmitrenok & I. V. Zavarzin

Authors
  1. L. S. Vasil’ev
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  2. S. V. Baranin
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  3. A. S. Dmitrenok
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  4. I. V. Zavarzin
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Corresponding author

Correspondence to S. V. Baranin.

Additional information

Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 9, pp. 1795–1797, September, 2019.

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Vasil’ev, L.S., Baranin, S.V., Dmitrenok, A.S. et al. A new approach to CF3-containing 3,4-dihydroquinazolin-2(1H)-ones. Russ Chem Bull 68, 1795–1797 (2019). https://doi.org/10.1007/s11172-019-2627-8

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  • DOI: https://doi.org/10.1007/s11172-019-2627-8

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