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Synthesis of succinic monoamide avermectin esters

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Abstract

Reaction of avermectin B1 hemisuccinate with N-hydroxysuccinimide and N,N’-dicyclohexylcarbodiimide followed by amination provided succinic monoamide avermectine esters that are potential antiparasitics.

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Authors and Affiliations

  1. N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991, Moscow, Russian Federation

    M. A. Shchetinina, E. I. Chernoburova, N. G. Kolotyrkina & I. V. Zavarzin

  2. K. I. Skryabin Moscow State Academy of Veterinary Medicine and Biotechnology, 23 ul. Akad. Skryabina, 109472, Moscow, Russian Federation

    M. Kh. Dzhafarov & F. I. Vasilevich

Authors
  1. M. A. Shchetinina
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  2. E. I. Chernoburova
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  3. N. G. Kolotyrkina
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  4. M. Kh. Dzhafarov
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  5. F. I. Vasilevich
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  6. I. V. Zavarzin
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Corresponding author

Correspondence to I. V. Zavarzin.

Additional information

Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 5, pp. 1116–1121, May, 2019.

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Shchetinina, M.A., Chernoburova, E.I., Kolotyrkina, N.G. et al. Synthesis of succinic monoamide avermectin esters. Russ Chem Bull 68, 1116–1121 (2019). https://doi.org/10.1007/s11172-019-2528-x

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  • DOI: https://doi.org/10.1007/s11172-019-2528-x

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