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Synthesis of ivermectin-4″,5-diyl[bis(N-methylcarbamate)]

Russian Chemical Bulletin volume 67, pages 833–835 (2018)Cite this article

Abstract

New ivermectin-4″,5-diyl[bis(N-methylcarbamate)] was synthesized by the MoO2Cl2(DMF)2-catalyzed reaction of ivermectin with methyl isocyanate. The synthesized compound could find application as antiparasitic agent.

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Authors and Affiliations

  1. N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991, Moscow, Russian Federation

    A. N. Blinnikov, E. I. Chernoburova, N. G. Kolotyrkina, M. A. Shchetinina & I. V. Zavarzin

  2. K. I. Skryabin Moscow State Academy of Veterinary Medicine and Biotechnology, 23 ul. Akad. Skryabina, 109472, Moscow, Russian Federation

    V. A. Lishchuk, K. L. Ovchinnikov, A. V. Kolobov, M. Kh. Dzhafarov & F. I. Vasilevich

Authors
  1. A. N. Blinnikov
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  2. E. I. Chernoburova
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  3. N. G. Kolotyrkina
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  4. M. A. Shchetinina
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  5. V. A. Lishchuk
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  6. K. L. Ovchinnikov
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  7. A. V. Kolobov
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  8. M. Kh. Dzhafarov
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  9. F. I. Vasilevich
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  10. I. V. Zavarzin
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Corresponding author

Correspondence to I. V. Zavarzin.

Additional information

Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 5, pp. 0833–0835, May, 2018.

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Blinnikov, A.N., Chernoburova, E.I., Kolotyrkina, N.G. et al. Synthesis of ivermectin-4″,5-diyl[bis(N-methylcarbamate)]. Russ Chem Bull 67, 833–835 (2018). https://doi.org/10.1007/s11172-018-2145-0

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  • DOI: https://doi.org/10.1007/s11172-018-2145-0

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