Abstract
7-Aryl- and 7-alkyl-6,7-dihydro-4H-thiazolo[4,5-b]pyridin-5-ones were obtained by three-component condensation of 5-unsubstituted 2-amino-4-iminothiazolidine hydrochlorides with aromatic or aliphatic aldehydes and Meldrum’s acid.
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Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 8, pp. 1707–1710, August, 2008.
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Dudinov, A.A., Lichitsky, B.V., Antonov, I.A. et al. Three-component condensation of 2,4-diaminothiazoles with aldehydes and Meldrum’s acid. The synthesis of 7-aryl- and 7-alkyl-6,7-dihydro-4H-thiazolo[4,5-b]pyridin-5-ones. Russ Chem Bull 57, 1740–1743 (2008). https://doi.org/10.1007/s11172-008-0230-5
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DOI: https://doi.org/10.1007/s11172-008-0230-5