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Conjugates of polyhedral boron compounds with carbohydrates

5. Synthesis of glycoconjugates of closo-ortho-carborane and N-acyl-β-lactosylamines with various spacers

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Russian Chemical Bulletin Aims and scope

Abstract

Conjugates of β-lactosylamine derivatives bearing terminal amino groups in aglycon with ortho-carboranylacetic acid were synthesized. Five glycoconjugates with spacers of different length (from 9 to 18 atoms) and hydrophilicity containing di-, tri-, and pentapeptide fragments constructed of glycine and serine residues and spacers incorporating ethylenediamine and tartaric acid or tertiary amine residues were prepared

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Authors and Affiliations

  1. N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991, Moscow, Russian Federation

    L. M. Likhosherstov, O. S. Novikova, L. O. Kononov & A. V. Orlova

  2. A. N. Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, 28 ul. Vavilova, 119991, Moscow, Russian Federation

    I. B. Sivaev & V. I. Bregadze

Authors
  1. L. M. Likhosherstov
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  2. O. S. Novikova
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  3. L. O. Kononov
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  4. A. V. Orlova
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  5. I. B. Sivaev
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  6. V. I. Bregadze
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Corresponding author

Correspondence to L. O. Kononov.

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Dedicated to the memory of outstanding chemist and biochemist V. N. Shibaev.

Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 10, pp. 2033–2036, October, 2007.

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Likhosherstov, L.M., Novikova, O.S., Kononov, L.O. et al. Conjugates of polyhedral boron compounds with carbohydrates. Russ Chem Bull 56, 2105–2108 (2007). https://doi.org/10.1007/s11172-007-0328-1

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  • DOI: https://doi.org/10.1007/s11172-007-0328-1

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