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Structural Features and Anti-Inflammatory Activity of 13-(N-Arylaminocarbonyl)-9-Methyl-11-Thioxo-8-Oxa-10,12-Diazatricyclo-[7.3.1.02,7]Trideca-2,4,6-Trienes and Their 10-N-Phenyl-Substituted Derivatives

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Pharmaceutical Chemistry Journal Aims and scope

A study of the structural features and anti-inflammatory activity of 13-(N-arylaminocarbonyl)-9-methyl-11-thioxo-8-oxa-10,12-diazatricyclo[7.3.1.02,7]trideca-2,4,6-trienes and their N-phenyl-substituted derivatives revealed that these compounds exhibited high anti-inflammatory activity and could be rated as promising nonsteroidal anti-inflammatory drugs.

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Correspondence to N. A. Buzmakova.

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Translated from Khimiko-Farmatsevticheskii Zhurnal, Vol. 56, No. 12, pp. 44 – 46, December, 2022.

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Buzmakova, N.A., Zamaraeva, T.M., Rudakova, I.P. et al. Structural Features and Anti-Inflammatory Activity of 13-(N-Arylaminocarbonyl)-9-Methyl-11-Thioxo-8-Oxa-10,12-Diazatricyclo-[7.3.1.02,7]Trideca-2,4,6-Trienes and Their 10-N-Phenyl-Substituted Derivatives. Pharm Chem J 56, 1613–1615 (2023). https://doi.org/10.1007/s11094-023-02835-y

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