Pharmaceutical Chemistry Journal

, Volume 49, Issue 1, pp 21–23 | Cite as

Synthesis, Protistocidal and Antibacterial Activities of 2′-Imidazolinylhydrazones of Mono- and Dicarboxylic Acids

  • L. D. Popov
  • S. I. Levchenkov
  • A. A. Zubenko
  • I. N. Shcherbakov
  • L. N. Fetisov
  • A. N. Bodryakov
  • O. V. Maevskii
  • V. A. Kogan
Article

We report here the synthesis of a series of imidazolinylhydrazones of salicylaldehyde and their substituted 2-N-tosylaminobenzaldehyde, 2-diphenylphosphinobenzaldehyde, and diacetylmonooxime derivatives, as well as the bis-imidazolinylhydrazones of 2,6-diformyl-4-tert-butylphenol and 2,6-diacetylpyridine. The protistocidal and antibacterial activities of the compounds made here were studied, and some were found to have high levels of protistocidal activity.

Keywords

imidazolinylhydrazones synthesis protistocide antibacterial activity 

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Copyright information

© Springer Science+Business Media New York 2015

Authors and Affiliations

  • L. D. Popov
    • 1
  • S. I. Levchenkov
    • 2
  • A. A. Zubenko
    • 3
  • I. N. Shcherbakov
    • 1
  • L. N. Fetisov
    • 3
  • A. N. Bodryakov
    • 3
  • O. V. Maevskii
    • 1
  • V. A. Kogan
    • 1
  1. 1.Southern Federal UniversityRostov-on-DonRussia
  2. 2.Southern Scientific CenterRussian Academy of SciencesRostov-on-DonRussia
  3. 3.North Caucasus Zonal Science Research Veterinary InstituteNovocherkasskRussia

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