Quinoline-Thioureidopeptides: A New Approach for the Synthesis of Quinoline-Isothiocyanate and Their Peptide Linkage
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We present an efficient synthetic route for quinoline condensed thioureidopeptidyl esters from corresponding isothiocyanate and amino acid esters. The utility of quinoline isothiocyanate as major building block for desired thioureidopeptides of quinoline interests, with good yield with excellent purity. All the new compounds are well characterized by IR, 1H NMR, mass and elemental analysis data.
KeywordsQuinoline-thioureidopeptides Isothiocyanate Amino acid ester
We thank to Kuvempu University for providing JRF, Indian Institute of science, Bangalore, for providing spectral data and University of Mysore, for providing elemental analysis facility.
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