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Synthesis of lappaconitine N-oxide under microwave activation

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Chemistry of Heterocyclic Compounds Aims and scope

Lappaconitine N-oxide was obtained in high yield via oxidation of lappaconitine with Oxone® in H2O–MeCN media under the conditions of microwave activation.

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Authors and Affiliations

  1. N. N. Vorozhtsov Novosibirsk Institute of Organic Chemistry, 9 Academician Lavrientiev Ave.,, Novosibirsk, 630090, Russia

    Natalia A. Pankrushina

  2. Novosibirsk State University, 2 Pirogov St., Novosibirsk, 630090, Russia

    Kymbat B. Rakhmetali

Authors
  1. Natalia A. Pankrushina
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  2. Kymbat B. Rakhmetali
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Correspondence to Natalia A. Pankrushina.

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Translated from Khimiya Geterotsiklicheskikh Soedinenii, 2016, 52(11), 970–972

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Pankrushina, N.A., Rakhmetali, K.B. Synthesis of lappaconitine N-oxide under microwave activation. Chem Heterocycl Comp 52, 970–972 (2016). https://doi.org/10.1007/s10593-017-1995-y

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  • DOI: https://doi.org/10.1007/s10593-017-1995-y

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